SCHEMBL7212988

SCHEMBL7212988

NC(=O)C1OC(CCCO)CC1(NS(=O)(=O)c1ccc(OCc2ccc(Cl)cc2F)cc1)C(=O)O

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MMP1 P03956 8/20 0.41
ADAM17 P78536 5/20 0.41
MMP13 P45452 5/20 0.37
ADAMTS5 Q9UNA0 5/20 0.37
ADAMTS7 Q9UKP4 1/20 0.37
ADAMTS4 O75173 4/20 0.36
MMP2 P08253 3/20 0.36
MMP14 P50281 2/20 0.36
MMP3 P08254 1/20 0.36
MMP9 P14780 1/20 0.36
MMP12 P39900 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7214339 0.91 MMP1 (0.40) MMP1ADAM17MMP13ADAMTS5ADAMTS7
SCHEMBL7214304 0.88 MMP1 (0.37) MMP1ADAM17MMP13ADAMTS5ADAMTS7
SCHEMBL7212996 0.88 MMP1 (0.42) MMP1ADAM17MMP13ADAMTS5ADAMTS7
SCHEMBL7209169 0.84 MMP1 (0.43) MMP1ADAM17MMP13ADAMTS5ADAMTS7
SCHEMBL7213084 0.84 ADAMTS5 (0.40) MMP1ADAM17MMP13ADAMTS5ADAMTS7
SCHEMBL7208577 0.81 ADAM17 (0.39) MMP1ADAM17MMP13ADAMTS5ADAMTS7
SCHEMBL7212982 0.81 ADAMTS5 (0.47) MMP1ADAM17MMP13ADAMTS5ADAMTS7
SCHEMBL7208604 0.78 ADAMTS5 (0.47) MMP1ADAM17MMP13ADAMTS5ADAMTS7
SCHEMBL7212985 0.78 MMP1 (0.51) MMP1ADAM17MMP13ADAMTS5ADAMTS7
SCHEMBL7207012 0.76 MMP13 (0.49) MMP1ADAM17MMP13ADAMTS5ADAMTS7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1181285-B1 3-(ARYLSULFONYLAMINO)-TETRAHYDROFURAN-3-CARBOXYLIC ACID HYDROXAMIDES PFIZER PROD INC (US) 2003-10-08 EP disclosed
EP-1181285-A2 3-(ARYLSULFONYLAMINO)-TETRAHYDROFURAN-3-CARBOXYLIC ACID HYDROXAMIDES Pfizer Products Inc. (US) 2002-02-27 EP disclosed
US-6342521-B1 DRUGS FOR TREATMENT OF ARTHRITIS PFIZER INC. 2002-01-29 US disclosed
WO-2000073294-A2 3-(ARYLSULFONYLAMINO)-TETRAHYDROFURAN-3-CARBOXYLIC ACID HYDROXAMIDES PFIZER PRODUCTS INC. (US) 2000-12-07 WO disclosed