SCHEMBL7208689

SCHEMBL7208689

O=S(=O)(CCCS)c1ccccc1Oc1ccccc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP8 P22894 4/20 0.63
MMP13 P45452 4/20 0.63
MMP3 P08254 3/20 0.63
MMP1 P03956 1/20 0.63
CASP1 P29466 1/20 0.41
MMP2 P08253 2/20 0.40
MMP9 P14780 2/20 0.40
MMP14 P50281 1/20 0.40
HDAC3 O15379 3/20 0.39
HDAC4 P56524 3/20 0.39
HDAC1 Q13547 3/20 0.39
HDAC7 Q8WUI4 3/20 0.39
HDAC2 Q92769 3/20 0.39
HDAC10 Q969S8 3/20 0.39
HDAC11 Q96DB2 3/20 0.39
HDAC8 Q9BY41 3/20 0.39
HDAC6 Q9UBN7 3/20 0.39
HDAC9 Q9UKV0 3/20 0.39
HDAC5 Q9UQL6 3/20 0.39
RIPK1 Q13546 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18184670 0.78 RIPK1 (0.47) CASP1RIPK1SLC6A2SLC6A4LMNA
SCHEMBL7208687 0.78 MMP13 (1.00) MMP8MMP13MMP3MMP1MMP2
SCHEMBL12748077 0.74 MMP8 (0.75) MMP8MMP13MMP3MMP1MMP2
SCHEMBL146565 0.74 CASP1 (0.50) MMP8MMP13MMP3CASP1MMP2
SCHEMBL502864 0.74 CASP1 (0.50) MMP8MMP13MMP3CASP1MMP2
SCHEMBL17038517 0.73 CASP1 (0.42) MMP13CASP1MMP2RIPK1LMNA
SCHEMBL7212096 0.72 MMP8 (0.47) MMP8MMP13MMP3MMP1CASP1
SCHEMBL11599660 0.72 CASP1 (0.49) MMP8MMP13MMP3CASP1MMP2
Ammonia Solution, Strong SCHEMBL502557 0.72 CASP1 (0.49) MMP8MMP13MMP3CASP1MMP2
SCHEMBL569758 0.71 SOS1 (0.55) CASP1LMNAGAAKMT2APTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0939628-B1 THIOL SULFONE METALLOPROTEASE INHIBITORS MONSANTO CO (US) 2003-03-05 EP disclosed
US-6013649-A BOND DISORDERS; AUTOIMMUNE DISEASES; ANTITUMOR AGENTS MONSANTO COMPANY (US) 2000-01-11 US disclosed
EP-0939628-A4 THIOL SULFONE METALLOPROTEASE INHIBITORS MONSANTO CO (US) 1999-12-22 EP disclosed
EP-0939628-A1 THIOL SULFONE METALLOPROTEASE INHIBITORS MONSANTO COMPANY (US) 1999-09-08 EP disclosed
WO-1998003164-A1 THIOL SULFONE METALLOPROTEASE INHIBITORS MONSANTO COMPANY (US) 1998-01-29 WO disclosed