SCHEMBL7215330

SCHEMBL7215330

Cc1c(Sc2ccccc2)n(C)c(=O)[nH]c1=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.43
LMNA P02545 2/20 0.43
PKM P14618 1/20 0.43
TSHR P16473 1/20 0.43
MAPK1 P28482 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
DRD1 P21728 2/20 0.38
GFER P55789 1/20 0.38
GAA P10253 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
KMT2A Q03164 1/20 0.37
ADORA3 P0DMS8 1/20 0.37
ADORA2A P29274 1/20 0.37
ADORA2B P29275 1/20 0.37
ADORA1 P30542 1/20 0.37
MAPT P10636 1/20 0.36
HPGD P15428 2/20 0.36
KDM4E B2RXH2 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7218800 0.78 ALDH1A1 (0.38) ALDH1A1LMNAPKMTSHRMAPK1
SCHEMBL7213302 0.77 MAPK1 (0.44) ALDH1A1LMNAPKMTSHRMAPK1
SCHEMBL7215341 0.77 ALDH1A1 (0.44) ALDH1A1LMNAPKMTSHRMAPK1
SCHEMBL8770174 0.74 UPP1 (0.42) ALDH1A1LMNAPKMTSHRMAPK1
SCHEMBL7015162 0.74 ALDH1A1 (0.58) ALDH1A1LMNAPKMTSHRMAPK1
SCHEMBL7260701 0.73 LMNA (0.37) ALDH1A1LMNAPKMTSHRMAPK1
Hept SCHEMBL384288 0.72 UPP1 (0.48) ALDH1A1TSHRMAPK1NPSR1CYP2C9
SCHEMBL14439983 0.71 ALDH1A1 (0.39) ALDH1A1LMNAPKMTSHRMAPK1
SCHEMBL7260700 0.70 ALDH1A1 (0.36) ALDH1A1LMNAPKMTSHRMAPK1
SCHEMBL7219572 0.69 ALDH1A1 (0.39) ALDH1A1TSHRMAPK1NPSR1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070190523-A1 Method and compositions for identifying anti-hiv therapeutic compounds GILEAD SCIENCES, INC. 2007-08-16 US disclosed
US-RE37979-E1 Pyrimidine derivatives and anti-viral agent containing the same as active ingredient thereof MITSUBISHI CHEMICAL CORPORATION 2003-02-04 US disclosed
EP-0829476-B1 6-Substituted acyclopyrimidine nucleoside derivatives and antiviral agent containing the same as active ingredient thereof MITSUBISHI CHEM CORP (JP) 2002-08-28 EP disclosed
EP-0829476-A2 6-Substituted acyclopyrimidine nucleoside derivatives and antiviral agent containing the same as active ingredient thereof Mitsubishi Chemical Corporation (JP) 1998-03-18 EP disclosed
US-5461060-A Antiretroviral activity MITSUBISHI KASEI CORPORATION (JP) 1995-10-24 US disclosed
EP-0420763-A2 6-Substituted acyclopyrimidine nucleoside derivatives and antiviral agent containing the same as active ingredient thereof Mitsubishi Chemical Corporation (JP) 1991-04-03 EP disclosed