SCHEMBL7215386

SCHEMBL7215386

CN(C)c1cc(-c2ccnc(S(C)(=O)=O)n2)c(-c2cccc(C(F)(F)F)c2)nn1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK11 Q15759 11/20 0.61
MAPK14 Q16539 11/20 0.61
MAPK13 O15264 9/20 0.61
MAPK12 P53778 9/20 0.61
MAOB P27338 1/20 0.40
KMO O15229 1/20 0.40
MAPK9 P45984 1/20 0.40
CSNK1D P48730 2/20 0.38
MAOA P21397 2/20 0.38
SDHB P21912 2/20 0.38
MEN1 O00255 1/20 0.38
S1PR4 O95977 1/20 0.38
LMNA P02545 1/20 0.38
TP53 P04637 1/20 0.38
POLB P06746 1/20 0.38
HPGD P15428 1/20 0.38
S1PR1 P21453 1/20 0.38
MAPK1 P28482 1/20 0.38
STAT3 P40763 1/20 0.38
STAT1 P42224 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7001627 0.87 MAPK13 (0.50) MAPK11MAPK14MAPK13MAPK12MAOB
SCHEMBL7215845 0.82 MAPK14 (0.63) MAPK11MAPK14MAPK13MAPK12MAOB
SCHEMBL17590 0.81 KMO (0.59) MAOBKMOSDHBMEN1S1PR4
SCHEMBL7676169 0.80 KMO (0.47) MAPK11MAPK14MAPK13MAPK12MAOB
SCHEMBL7215944 0.79 MAPK13 (0.65) MAPK11MAPK14MAPK13MAPK12MAPK9
SCHEMBL1384726 0.78 TGFBR1 (0.41) MAPK11MAPK14MAPK13MAPK12KMO
SCHEMBL7215839 0.75 MAPK14 (0.69) MAPK11MAPK14MAPK13MAPK12MAPK9
SCHEMBL14561097 0.72 MAPT (0.44) MAPK11MAPK14MAPK13MAPK12KMO
SCHEMBL14561100 0.72 BRAF (0.50) MAPK11MAPK14KMOSDHBMEN1
SCHEMBL5823023 0.72 CDC7 (0.44) MAPK14KMOSDHBMEN1S1PR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6602872-B1 Substituted pyridazines having cytokine inhibitory activity MERCK & CO., INC. 2003-08-05 US disclosed