SCHEMBL7216137

SCHEMBL7216137

Cc1c(-c2c[nH]c(NC(C)c3ccc(Cl)cc3)n2)ccc2ccccc12

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE9A O76083 6/20 0.37
GRK6 P43250 1/20 0.35
PDE5A O76074 2/20 0.34
PDE1B Q01064 2/20 0.34
PDE2A O00408 1/20 0.34
PDE8A O60658 1/20 0.34
PDE4D Q08499 1/20 0.34
PDE7A Q13946 1/20 0.34
PDE10A Q9Y233 1/20 0.34
ATP1A1 P05023 1/20 0.34
ATP1B1 P05026 1/20 0.34
ATP1A3 P13637 1/20 0.34
ATP1B2 P14415 1/20 0.34
ATP1A2 P50993 1/20 0.34
ATP1B3 P54709 1/20 0.34
FXYD2 P54710 1/20 0.34
ATP1A4 Q13733 1/20 0.34
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
LDHA P00338 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7217987 0.89 CCNE2 (0.40) GRK6ATP1A1ATP1B1ATP1A3ATP1B2
SCHEMBL7221634 0.86 ATP1A1 (0.37) ATP1A1ATP1B1ATP1A3ATP1B2ATP1A2
SCHEMBL7215523 0.85 SOS1 (0.37) MAPTNPSR1GAAKMT2AAR
SCHEMBL7222409 0.79 APP (0.39) PDE5AMAPTKMT2AHSD17B10
SCHEMBL7215731 0.77 KMT2A (0.35) MAPTNPSR1KDM4EGAAKMT2A
SCHEMBL7222469 0.75 CDK2 (0.34) SLC6A2SLC6A4MAPTHPGDNPSR1
SCHEMBL7216330 0.73 CD38 (0.40) PDE9AMAPTCYP3A4CYP2C9KMT2A
SCHEMBL7215977 0.67 NTRK1 (0.39) GRK6MAPTHPGDKDM4EGAA
SCHEMBL7216134 0.67 ATP1A1 (0.48) PDE9APDE1BATP1A1ATP1B1ATP1A3
SCHEMBL28676692 0.63 GAA (0.61) ATP1A1ATP1B1ATP1A3ATP1B2ATP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6596739-B2 Anticarcinogenic agents, cardiovascular disorders and antiinflammatory agents THE PROCTER & GAMBLE COMPANY 2003-07-22 US claimed