SCHEMBL7217545

SCHEMBL7217545

CC(C)c1[nH]cc(-c2ccccc2)c1-c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.40
ALDH1A1 P00352 1/20 0.39
HTT P42858 1/20 0.36
GCGR P47871 1/20 0.35
GRM5 P41594 2/20 0.35
ADRA2A P08913 1/20 0.35
ADRA2B P18089 1/20 0.35
ADRA2C P18825 1/20 0.35
CDK8 P49336 2/20 0.34
LRRK2 Q5S007 2/20 0.34
AXL P30530 1/20 0.34
TNIK Q9UKE5 1/20 0.34
METAP2 P50579 1/20 0.34
ADORA3 P0DMS8 1/20 0.34
ADORA2A P29274 1/20 0.34
ADORA2B P29275 1/20 0.34
ADORA1 P30542 1/20 0.34
CDC25A P30304 1/20 0.33
CDC25B P30305 1/20 0.33
PRKD3 O94806 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27577761 0.75 HTT (0.49) PARP1ALDH1A1HTTADRA2BAXL
SCHEMBL9459084 0.74 HTT (0.50) PARP1ALDH1A1HTTGRM5CDK8
SCHEMBL13301396 0.72 MAPT (0.44) PARP1ALDH1A1ADRA2AADRA2BADRA2C
SCHEMBL4792528 0.71 PARP1 (0.45) PARP1ALDH1A1GRM5CDK8LRRK2
SCHEMBL29264066 0.69 LMNA (0.44) PARP1ALDH1A1HTTGRM5CDK8
SCHEMBL12912923 0.69 PARP1 (0.44) PARP1ALDH1A1HTTGRM5CDK8
Hydrochloric Acid SCHEMBL28338871 0.69 CHEK1 (0.44) PARP1ALDH1A1GRM5CDK8LRRK2
SCHEMBL12912920 0.69 ALDH1A1 (0.43) PARP1ALDH1A1HTTGRM5CDK8
SCHEMBL12912922 0.69 CDK8 (0.41) PARP1ALDH1A1HTTGRM5CDK8
SCHEMBL1127324 0.69 HTT (0.46) PARP1ALDH1A1HTTCDK8LRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6590119-B2 Catalytic alcoholysis of benzoylcyclohexanone ketals; products useful as intermediates for diarylpyrrole therapeutic agents ORTHO-MCNEIL PHARMACEUTICAL, INC. 2003-07-08 US disclosed
US-20020107408-A1 Methods for the synthesis of dioxoalkanoic acid compounds FERRO MICHAEL P (US) 2002-08-08 US disclosed
US-6355812-B1 ALCOHOLYSIS OF BENZOYLCYCLOHEXANONE KETAL COMPOUNDS ORTH-MCNEIL PHARMACEUTICAL, INC. 2002-03-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020107408-A1 Methods for the synthesis of dioxoalkanoic acid compounds DCK, DDT, AOX1 PARP1 1164/4885ALDH1A1 281/4885HTT 1173/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.