SCHEMBL7223372

SCHEMBL7223372

Cc1nc(C(=O)N[C@@H]2C[C@H]3CC[C@@H]2N3)sc1-c1ccccc1F

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 1/20 0.36
PIK3CD O00329 1/20 0.36
PIK3CA P42336 1/20 0.36
KDM1A O60341 1/20 0.36
HCRTR1 O43613 2/20 0.35
HCRTR2 O43614 2/20 0.35
TSPO P30536 1/20 0.35
OPRK1 P41145 1/20 0.35
HTR2B P41595 1/20 0.35
FFAR4 Q5NUL3 1/20 0.35
CTSK P43235 1/20 0.34
CTSC P53634 1/20 0.34
SLC6A2 P23975 2/20 0.34
SLC6A4 P31645 2/20 0.34
SLC6A3 Q01959 2/20 0.34
HTR3E A5X5Y0 1/20 0.34
HTR3B O95264 1/20 0.34
HTR3A P46098 1/20 0.34
HTR3D Q70Z44 1/20 0.34
HTR3C Q8WXA8 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7230427 0.88 CNR1 (0.36) SLC6A2SLC6A4SLC6A3HTR3EHTR3B
SCHEMBL7223552 0.88 NPC1 (0.38) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL7232879 0.86 CHRM4 (0.41) KDM1AHCRTR1HCRTR2HTR3EHTR3B
SCHEMBL7224821 0.84 CTSK (0.37) HCRTR1HCRTR2CTSKCTSCSLC6A2
SCHEMBL7231066 0.82 KDM4E (0.39) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL7225526 0.82 DGAT1 (0.39) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL7230824 0.80 CHRNB2 (0.39) HCRTR1HCRTR2SLC6A3CHRNB2CHRNA4
SCHEMBL7233563 0.79 HCRTR1 (0.40) HCRTR1HCRTR2SLC6A2SLC6A4SLC6A3
SCHEMBL7075331 0.78 USP30 (0.39) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL7059395 0.77 CHRNA7 (0.54) HTR3EHTR3BHTR3AHTR3DHTR3C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US claimed
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US disclosed