SCHEMBL7232879

SCHEMBL7232879

COc1ccccc1-c1sc(C(=O)N[C@@H]2C[C@H]3CC[C@@H]2N3)nc1C

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CHRM4 P08173 1/20 0.41
CHRNA7 P36544 2/20 0.39
KDM1A O60341 1/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
HTR3A P46098 2/20 0.37
HTR3E A5X5Y0 1/20 0.37
HTR3B O95264 1/20 0.37
HTR3D Q70Z44 1/20 0.37
HTR3C Q8WXA8 1/20 0.37
HCRTR1 O43613 3/20 0.37
HCRTR2 O43614 2/20 0.37
FAAH O00519 1/20 0.36
CNR2 P34972 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7230427 0.86 CNR1 (0.36) CHRNA7NPC1RAB9AHTR3AHTR3E
SCHEMBL7223372 0.86 RIPK1 (0.36) KDM1AHTR3AHTR3EHTR3BHTR3D
SCHEMBL7223552 0.86 NPC1 (0.38) CHRNA7NPC1RAB9AHTR3AHTR3E
SCHEMBL7234242 0.83 HDAC3 (0.47) CHRNA7KDM1ANPC1RAB9AHTR3A
SCHEMBL7233563 0.83 HCRTR1 (0.40) NPC1RAB9AHCRTR1HCRTR2FAAH
SCHEMBL7231066 0.80 KDM4E (0.39) CHRNA7NPC1RAB9AHTR3AHTR3E
SCHEMBL7232275 0.79 CHRNA7 (0.62) CHRNA7HTR3AHTR3EHTR3BHTR3D
SCHEMBL7233270 0.79 HDAC3 (0.48) CHRNA7KDM1ANPC1RAB9AHTR3A
SCHEMBL7230824 0.79 CHRNB2 (0.39) NPC1RAB9AHCRTR1HCRTR2CNR2
SCHEMBL7224821 0.79 CTSK (0.37) HCRTR1HCRTR2FAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US claimed
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US disclosed