SCHEMBL7223387

SCHEMBL7223387

NS(=O)(=O)c1ccc(Oc2ccc(C(=O)N[C@@H]3C[C@H]4CC[C@@H]3N4)s2)cc1

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.35
HTT P42858 1/20 0.35
CHRNB2 P17787 1/20 0.34
CHRNA4 P43681 1/20 0.34
CA2 P00918 6/20 0.33
CA1 P00915 5/20 0.33
CA9 Q16790 3/20 0.33
CA12 O43570 2/20 0.33
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
SOS1 Q07889 2/20 0.32
CA4 P22748 2/20 0.31
CA7 P43166 2/20 0.31
MAPT P10636 2/20 0.31
SLC8A1 P32418 2/20 0.31
KDM4E B2RXH2 1/20 0.30
GAA P10253 1/20 0.30
POLB P06746 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7234327 0.89 KMT2A (0.36) CHRNB2CHRNA4MEN1KMT2ASLC8A1
SCHEMBL7232095 0.88 CHRNA7 (0.34) ALDH1A1SLC8A1
SCHEMBL7233323 0.87 ESR1 (0.37) ALDH1A1
SCHEMBL7224931 0.86 F2 (0.37) ALDH1A1CHRNB2CHRNA4KMT2A
SCHEMBL7225149 0.86 HTR4 (0.37) ALDH1A1MAPTKDM4EGAAPOLB
SCHEMBL7225066 0.86 SLC6A4 (0.41) CHRNB2CHRNA4KMT2AKDM4E
SCHEMBL7229845 0.86 SLC6A3 (0.42) POLB
SCHEMBL7225381 0.86 HTR3E (0.37)
SCHEMBL7232594 0.85 HTT (0.40) ALDH1A1HTTKDM4EGAA
SCHEMBL7231419 0.84 SCN9A (0.37) MEN1KMT2AMAPTKDM4EPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US claimed
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US disclosed