SCHEMBL7224405

SCHEMBL7224405

O=C(N[C@@H]1C[C@H]2CC[C@@H]1N2)c1ncc(Oc2ccccc2F)o1

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 4/20 0.36
HPGD P15428 1/20 0.35
SLC6A2 P23975 2/20 0.33
SLC6A4 P31645 2/20 0.33
KDM1A O60341 1/20 0.33
HTR3E A5X5Y0 1/20 0.33
HTR3B O95264 1/20 0.33
HTR3A P46098 1/20 0.33
HTR3D Q70Z44 1/20 0.33
HTR3C Q8WXA8 1/20 0.33
CHRNA1 P02708 1/20 0.33
CHRNG P07510 1/20 0.33
ITGA5 P08648 1/20 0.33
CHRNB1 P11230 1/20 0.33
CHRNB2 P17787 1/20 0.33
CHRNB4 P30926 1/20 0.33
CHRNA3 P32297 1/20 0.33
CHRNA4 P43681 1/20 0.33
CHRND Q07001 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7231938 0.91 MAPK14 (0.40) SLC6A3SLC6A2SLC6A4KDM1A
SCHEMBL7225396 0.89 SLC6A4 (0.37) SLC6A3SLC6A2SLC6A4HTR3EHTR3B
SCHEMBL7225383 0.86 SLC6A3 (0.41) SLC6A3
SCHEMBL7233162 0.86 HTR3E (0.38) SLC6A3SLC6A2SLC6A4HTR3EHTR3B
SCHEMBL7225309 0.84 PDE4A (0.35) SLC6A3SLC6A2SLC6A4KDM1ACHRNA1
SCHEMBL7230399 0.83 MAPT (0.36) SLC6A3HPGDSLC6A2SLC6A4KDM1A
SCHEMBL7231360 0.83 SLC6A3 (0.39) SLC6A3SLC6A2SLC6A4CHRNB2CHRNA4
SCHEMBL7234468 0.82 SLC6A3 (0.35) SLC6A3SLC6A2SLC6A4KDM1ACHRNA1
SCHEMBL7229511 0.81 FAAH (0.44) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL7231983 0.81 SLC6A3 (0.37) SLC6A3HPGDSLC6A2SLC6A4CHRNA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US claimed
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US disclosed