SCHEMBL7225396

SCHEMBL7225396

O=C(N[C@@H]1C[C@H]2CC[C@@H]1N2)c1ncc(Oc2ccccc2Cl)o1

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 5/20 0.37
SLC6A3 Q01959 5/20 0.37
SLC6A2 P23975 2/20 0.37
ABL1 P00519 1/20 0.35
EZH2 Q15910 1/20 0.33
HTR3E A5X5Y0 1/20 0.33
HTR3B O95264 1/20 0.33
HTR3A P46098 1/20 0.33
HTR3D Q70Z44 1/20 0.33
HTR3C Q8WXA8 1/20 0.33
CHRNA1 P02708 1/20 0.33
CHRNG P07510 1/20 0.33
ITGA5 P08648 1/20 0.33
CHRNB1 P11230 1/20 0.33
CHRNB2 P17787 1/20 0.33
CHRNB4 P30926 1/20 0.33
CHRNA3 P32297 1/20 0.33
CHRNA4 P43681 1/20 0.33
CHRND Q07001 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7231983 0.89 SLC6A3 (0.37) SLC6A4SLC6A3SLC6A2CHRNA1CHRNG
SCHEMBL7224405 0.89 SLC6A3 (0.36) SLC6A4SLC6A3SLC6A2HTR3EHTR3B
SCHEMBL7233162 0.86 HTR3E (0.38) SLC6A4SLC6A3SLC6A2HTR3EHTR3B
SCHEMBL7234091 0.84 SLC6A4 (0.41) SLC6A4SLC6A3SLC6A2CHRNB2CHRNB4
SCHEMBL7231538 0.84 SLC6A3 (0.42) SLC6A4SLC6A3SLC6A2CHRNA1CHRNG
SCHEMBL7232058 0.83 NPSR1 (0.40) SLC6A4SLC6A3SLC6A2EZH2
SCHEMBL7231938 0.83 MAPK14 (0.40) SLC6A4SLC6A3SLC6A2
SCHEMBL7223564 0.83 SLC6A4 (0.39) SLC6A4SLC6A3SLC6A2ABL1CHRNB2
SCHEMBL7232046 0.82 ALDH1A1 (0.39) SLC6A4SLC6A3SLC6A2CHRNA1CHRNG
SCHEMBL7225383 0.82 SLC6A3 (0.41) SLC6A3ABL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US claimed
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US disclosed