SCHEMBL7224822

SCHEMBL7224822

O=C(N[C@@H]1C[C@H]2CC[C@@H]1N2)c1ccc(-c2ccccn2)o1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 3/20 0.47
CHRNB2 P17787 1/20 0.47
CHRNA4 P43681 1/20 0.47
HSP90AA1 P07900 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
ALOX5 P09917 1/20 0.37
FAAH O00519 2/20 0.36
AKT1 P31749 1/20 0.36
GRM5 P41594 1/20 0.36
MDM4 O15151 1/20 0.36
MDM2 Q00987 1/20 0.36
HTR3E A5X5Y0 1/20 0.36
HTR3B O95264 1/20 0.36
HTR3A P46098 1/20 0.36
HTR3D Q70Z44 1/20 0.36
HTR3C Q8WXA8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7230688 0.85 AKT1 (0.44) CHRNA7CHRNB2CHRNA4L3MBTL1AKT1
SCHEMBL7224879 0.85 AKT1 (0.39) CHRNA7CHRNB2CHRNA4FAAHAKT1
SCHEMBL7231889 0.84 FAAH (0.49) FAAH
SCHEMBL7226398 0.84 AKT1 (0.34) CHRNA7CHRNB2CHRNA4L3MBTL1AKT1
SCHEMBL7232903 0.83 SLC6A3 (0.38) CHRNA7CHRNB2CHRNA4AKT1
SCHEMBL7232737 0.83 MMP13 (0.49) CHRNA7CHRNB2CHRNA4L3MBTL1AKT1
SCHEMBL7226388 0.83 AKT1 (0.37) CHRNA7CHRNB2CHRNA4L3MBTL1AKT1
SCHEMBL7074460 0.83 NPC1 (0.44) CHRNA7CHRNB2CHRNA4L3MBTL1
SCHEMBL375394 0.83 NPC1 (0.44) CHRNA7CHRNB2CHRNA4L3MBTL1
SCHEMBL7224807 0.82 MGAM (0.35) CHRNA7CHRNB2CHRNA4HSP90AA1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US claimed
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US disclosed