SCHEMBL7225781

SCHEMBL7225781

O=C(N[C@@H]1C[C@H]2CC[C@@H]1N2)c1ccc(Sc2cccc(Cl)c2)o1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PTPN11 Q06124 3/20 0.44
ATM Q13315 1/20 0.38
ALDH1A1 P00352 2/20 0.36
LMNA P02545 2/20 0.36
KDM4E B2RXH2 1/20 0.36
NPC1 O15118 1/20 0.36
MAPT P10636 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
GRM5 P41594 4/20 0.35
SLC6A4 P31645 2/20 0.34
SLC6A2 P23975 1/20 0.34
SLC6A3 Q01959 1/20 0.34
TP53 P04637 2/20 0.33
TRPV1 Q8NER1 1/20 0.33
CHRNB4 P30926 1/20 0.33
CHRNA3 P32297 1/20 0.33
THRB P10828 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7231968 0.88 ALDH1A1 (0.42) PTPN11ALDH1A1LMNAMAPTSMN1; SMN2
SCHEMBL7234113 0.88 PTPN11 (0.41) PTPN11ALDH1A1LMNAKDM4ENPC1
SCHEMBL7230851 0.88 CHRNA7 (0.35) ALDH1A1LMNASMN1; SMN2
SCHEMBL7224680 0.84 CHRNB2 (0.36) PTPN11GRM5SLC6A4SLC6A3
SCHEMBL7232031 0.83 PTPN11 (0.43) PTPN11ALDH1A1LMNANPC1RAB9A
SCHEMBL7225482 0.83 ALDH1A1 (0.54) ATMALDH1A1LMNAKDM4ENPC1
SCHEMBL7224259 0.82 SLC6A3 (0.39) ALDH1A1LMNAMAPTSMN1; SMN2SLC6A4
SCHEMBL7127459 0.82 CHRNA7 (0.43) NPC1RAB9AGRM5TRPV1
SCHEMBL7233643 0.80 NPC1 (0.41) ALDH1A1LMNAKDM4ENPC1MAPT
SCHEMBL7226375 0.79 MAPT (0.48) ATMALDH1A1LMNAKDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US claimed
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US disclosed