SCHEMBL7229190

SCHEMBL7229190

Cc1c(F)cc(-c2nc(NCC(N)=O)c(Cl)c(-c3ccccc3)n2)c(F)c1F

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 2/20 0.42
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
GAA P10253 1/20 0.41
IKBKB O14920 1/20 0.38
IRAK4 Q9NWZ3 1/20 0.37
LMNA P02545 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
NTRK1 P04629 2/20 0.35
PTGFR P43088 7/20 0.34
DHODH Q02127 2/20 0.34
CYP3A4 P08684 1/20 0.34
PRKCI P41743 1/20 0.33
ADK P55263 1/20 0.33
CDK1 P06493 1/20 0.32
CDK2 P24941 1/20 0.32
GSK3B P49841 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6946847 0.74 PDE10A (0.54) PDE10AKDM4EALDH1A1GAADHODH
SCHEMBL7230333 0.67 SYK (0.35) GAALMNASMN1; SMN2
SCHEMBL7077947 0.64 DHODH (0.40) KDM4EALDH1A1GAALMNADHODH
SCHEMBL7237373 0.63 POLB (0.34) LMNASMN1; SMN2
SCHEMBL718683 0.63 ALPL (0.34) KDM4EALDH1A1SMN1; SMN2
SCHEMBL5810835 0.61 PDE4B (0.61) PDE10AKDM4EALDH1A1GAALMNA
SCHEMBL7502850 0.59 MEN1 (0.59) PDE10AKDM4EALDH1A1GAASMN1; SMN2
SCHEMBL30009492 0.58 BCAT2 (0.49) IKBKBDHODH
SCHEMBL3253576 0.58 PDE10A (0.55) PDE10AKDM4EALDH1A1GAAIKBKB
SCHEMBL4516645 0.58 MEN1 (0.67) PDE10AALDH1A1GAALMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6620817-B1 Antiinflammatory, antiarthritic agents; autoimmune and rheumatic diseases DAINIPPON PHARMACEUTICAL CO., LTD. (JP) 2003-09-16 US claimed