SCHEMBL7231998

SCHEMBL7231998

COc1ccc(Oc2ccc(C(=O)N[C@@H]3C[C@H]4CC[C@@H]3N4)s2)cn1

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.35
CHRNA4 P43681 1/20 0.35
HTR4 Q13639 1/20 0.34
SCN9A Q15858 1/20 0.33
CTSC P53634 1/20 0.33
MMP3 P08254 1/20 0.33
MMP10 P09238 1/20 0.33
LMNA P02545 1/20 0.32
NPC1 O15118 1/20 0.32
POLB P06746 1/20 0.32
RAB9A P51151 1/20 0.32
MEN1 O00255 1/20 0.32
MAPT P10636 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7223716 0.93 SCN9A (0.35) HTR4SCN9ANPC1POLBRAB9A
SCHEMBL7231120 0.89 P2RY14 (0.38) CHRNB2CHRNA4
SCHEMBL7225892 0.88 CHRNB2 (0.39) CHRNB2CHRNA4NPC1RAB9AMEN1
SCHEMBL7225149 0.87 HTR4 (0.37) HTR4LMNANPC1POLBRAB9A
SCHEMBL7232573 0.86 CTSC (0.34) HTR4CTSCNPC1POLBRAB9A
SCHEMBL7225984 0.85 P2RY14 (0.37) SCN9ANPC1POLBRAB9A
SCHEMBL7224866 0.84 CTSC (0.40) CTSCLMNANPC1MAPT
SCHEMBL7116059 0.84 POLB (0.39) CHRNB2CHRNA4SCN9AMMP3MMP10
SCHEMBL7229845 0.83 SLC6A3 (0.42) NPC1POLBRAB9A
SCHEMBL7226161 0.83 SLC6A3 (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US claimed
US-6562816-B2 Alpha 7 nicotine acetylcholine receptor agonist anti-psychotic agent, with reduced side effects PHARMACIA & UPJOHN COMPANY 2003-05-13 US disclosed