SCHEMBL7236145

SCHEMBL7236145

C[SiH](C)Oc1c(C(C)(C)C)ccc([C@H](N)CC(=O)O)c1-c1ccccc1

nearest known ligand 0.34

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 1/20 0.34
PDE4A P27815 2/20 0.31
PDE4B Q07343 2/20 0.31
PDE4C Q08493 2/20 0.31
PDE4D Q08499 2/20 0.31
KMT2A Q03164 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
S1PR1 P21453 1/20 0.31
MMP12 P39900 1/20 0.30
FFAR1 O14842 1/20 0.30
RXRA P19793 1/20 0.30
RXRB P28702 1/20 0.30
RXRG P48443 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7622508 0.73 PDE4B (0.40) PDE4APDE4BPDE4CPDE4D
SCHEMBL7236273 0.70 CYP2C19 (0.39) SMN1; SMN2FFAR1RXRARXRBRXRG
Hydrochloric Acid SCHEMBL7236567 0.69 CYP2C19 (0.39) SMN1; SMN2FFAR1RXRARXRBRXRG
Hydrochloric Acid SCHEMBL7236577 0.69 CYP2C19 (0.39) SMN1; SMN2FFAR1RXRARXRBRXRG
SCHEMBL7236130 0.69 NPC1 (0.37)
SCHEMBL3235703 0.65 NR1H4 (0.43) MMP12RXRARXRBRXRG
SCHEMBL8675813 0.65 NPC1 (0.41) KMT2ASMN1; SMN2S1PR1
SCHEMBL27599721 0.63 L3MBTL1 (0.40) KMT2ASMN1; SMN2
SCHEMBL7714320 0.63 KMT2A (0.43) CASP1KMT2ASMN1; SMN2MMP12FFAR1
SCHEMBL2989103 0.62 ALDH1A1 (0.41) RXRARXRBRXRG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6645939-B1 Very late antigen-4 (VLA) integrin antagonists; antiallergens, antiasthmatics, and antiinflammatory agents; multiple sclerosis, autoimmune disease treatment MERCK & CO., INC. 2003-11-11 US disclosed