2,3,4-Trihydroxy-4'-Ethoxybenzophenone

2,3,4-Trihydroxy-4'-Ethoxybenzophenone

SCHEMBL724437

CCOc1ccc(C(=O)c2ccc(O)c(O)c2O)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 1.00
MAPT P10636 5/20 1.00
ALDH1A1 P00352 5/20 1.00
HPGD P15428 4/20 1.00
ALOX15 P16050 3/20 1.00
RECQL P46063 3/20 1.00
HSD17B10 Q99714 3/20 1.00
KMT2A Q03164 2/20 0.70
MEN1 O00255 1/20 0.70
ALOX12 P18054 1/20 0.70
NPSR1 Q6W5P4 2/20 0.54
PLK1 P53350 1/20 0.53
PARP10 Q53GL7 1/20 0.51
HDAC1 Q13547 1/20 0.51
MAPK1 P28482 3/20 0.50
TDP1 Q9NUW8 2/20 0.50
POLB P06746 1/20 0.50
HCRTR1 O43613 1/20 0.49
HCRTR2 O43614 1/20 0.49
NPC1 O15118 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29092709 0.88 KDM4E (0.78) KDM4EMAPTALDH1A1HPGDALOX15
SCHEMBL28998878 0.88 KDM4E (0.78) KDM4EMAPTALDH1A1HPGDALOX15
SCHEMBL29415000 0.86 KDM4E (0.84) KDM4EMAPTALDH1A1HPGDALOX15
SCHEMBL28137387 0.86 KDM4E (0.84) KDM4EMAPTALDH1A1HPGDALOX15
2,3-Dihydroxy-4-Methoxy-4'-Ethoxybenzophenone SCHEMBL4007549 0.84 MAPT (1.00) KDM4EMAPTALDH1A1HPGDALOX15
SCHEMBL29415019 0.83 KDM4E (0.70) KDM4EMAPTALDH1A1HPGDALOX15
SCHEMBL2488063 0.83 KDM4E (0.70) KDM4EMAPTALDH1A1HPGDALOX15
3,4-Didesmethyl-5-Deshydroxy-3'-Ethoxyscleroin SCHEMBL12998336 0.82 HPGD (1.00) KDM4EMAPTALDH1A1HPGDALOX15
SCHEMBL93601 0.82 MAPT (0.69) KDM4EMAPTALDH1A1HPGDALOX15
SCHEMBL18127697 0.82 ALDH1A1 (0.69) KDM4EMAPTALDH1A1HPGDALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 40 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20150044193-A1 COMPOSITIONS AND METHODS FOR THE TREATMENT OF ALTERED a-SYNUCLEIN FUNCTION NEURALTUS PHARMACEUTICALS, INC. 2015-02-12 US claimed
US-8669048-B2 Pluripotent cell lines and methods of use thereof PARKINSON'S INSTITUTE (US) 2014-03-11 US claimed
US-20120052053-A1 COMPOSITIONS AND METHODS FOR THE TREATMENT OF ALTERED ALPHA-SYNUCLEIN FUNCTION THE PARKINSON'S INSTITUTE 2012-03-01 US claimed
EP-2361089-A1 COMPOSITIONS AND METHODS FOR THE TREATMENT OF ALTERED -SYNUCLEIN FUNCTION Parkinson's Institute (US) 2011-08-31 EP claimed
US-20110189310-A1 SMALL MOLECULE MODULATORS OF PRONGF UPTAKE CORNELL UNIVERSITY (US) 2011-08-04 US claimed
US-20100167286-A1 Pluripotent cell lines and methods of use thereof PARKINSON'S INSTITUTE (US) 2010-07-01 US claimed
WO-2010056413-A2 COMPOSITIONS AND METHODS FOR THE TREATMENT OF ALTERED α-SYNUCLEIN FUNCTION PARKINSON'S INSTITUTE (US) 2010-05-20 WO claimed
WO-2010008486-A2 PLURIPOTENT CELL LINES AND METHODS OF USE THEREOF PARKINSONS INSTITUTE (US) 2010-01-21 WO claimed
US-10233422-B2 Pluripotent cell lines and methods of use thereof PARKINSON'S INSTITUTE (US) 2019-03-19 US disclosed
US-20180042899-A1 Method of Treating Transplant Rejection and Autoimmune Diseases NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2018-02-15 US disclosed
US-20170114324-A1 PLURIPOTENT CELL LINES AND METHODS OF USE THEREOF TYLER MEDICAL RESEARCH, LLC 2017-04-27 US disclosed
US-9527878-B2 Plasminogen activator inhibitor-1 inhibitors and methods of use thereof to modulate lipid metabolism THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2016-12-27 US disclosed
US-9527878-B2 Plasminogen activator inhibitor-1 inhibitors and methods of use thereof to modulate lipid metabolism THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2016-12-27 US disclosed
US-9527878-B2 Plasminogen activator inhibitor-1 inhibitors and methods of use thereof to modulate lipid metabolism THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2016-12-27 US disclosed
WO-2010042728-A1 SMALL MOLECULE MODULATORS OF PRONGF UPTAKE CORNELL UNIVERSITY (US) 2010-04-15 WO disclosed
WO-2010008486-A2 PLURIPOTENT CELL LINES AND METHODS OF USE THEREOF PARKINSONS INSTITUTE (US) 2010-01-21 WO disclosed
WO-2009081141-A1 BENZOPHENONE COMPOUNDS UNIVERSITY OF SHEFFIELD (GB) 2009-07-02 WO disclosed
WO-2009081141-A1 BENZOPHENONE COMPOUNDS UNIVERSITY OF SHEFFIELD (GB) 2009-07-02 WO disclosed
US-20090143279-A1 Methods and compositions for treating metabolic disorders PRESIDENT AND FELLOWS OF HARVARD COLLEGE 2009-06-04 US disclosed
WO-2009003147-A1 METHODS AND COMPOSITIONS FOR THE TREATMENT OF NEUROLOGICAL DISORDERS PARKINSON'S INSTITUTE (US) 2008-12-31 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120052053-A1 COMPOSITIONS AND METHODS FOR THE TREATMENT OF ALTERED ALPHA-SYNUCLEIN FUNCTION SNCA, PARK7, NLN KDM4E 4389/4885MAPT 55/4885ALDH1A1 2223/4885
US-20150044193-A1 COMPOSITIONS AND METHODS FOR THE TREATMENT OF ALTERED a-SYNUCLEIN FUNCTION SNCA, PARK7, NLN KDM4E 4335/4885MAPT 69/4885ALDH1A1 2054/4885
US-20090143279-A1 Methods and compositions for treating metabolic disorders PC, PCK2, CS KDM4E 3739/4885MAPT 357/4885ALDH1A1 860/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.