Bromide

Bromide

SCHEMBL7245264

O=S(=O)(NC(CC[P+](c1ccccc1)(c1ccccc1)c1ccccc1)Cc1ccccc1)c1ccccc1.[Br-]

nearest known ligand 0.56

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHECHKACHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGHRH2OPRM1

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 1/20 0.56
CA2 P00918 2/20 0.51
CA7 P43166 2/20 0.51
ALDH1A1 P00352 2/20 0.48
CYP1A2 P05177 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48
CTSL P07711 1/20 0.46
CTSS P25774 1/20 0.46
MMP2 P08253 8/20 0.45
MMP9 P14780 5/20 0.45
ADAMTS4 O75173 1/20 0.45
CA9 Q16790 2/20 0.44
CA1 P00915 1/20 0.44
CA4 P22748 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.43
HIF1A Q16665 1/20 0.43
LMTK3 Q96Q04 2/20 0.42
CA12 O43570 1/20 0.42
CA14 Q9ULX7 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL7245256 1.00 PIN1 (0.56) PIN1CA2CA7ALDH1A1CYP1A2
SCHEMBL7246631 0.81 PIN1 (0.57) PIN1CA2CA7ALDH1A1CYP1A2
SCHEMBL7246633 0.81 PIN1 (0.57) PIN1CA2CA7ALDH1A1CYP1A2
Bromide SCHEMBL27546307 0.79 PIN1 (0.56) PIN1CA2CA7ALDH1A1CYP1A2
SCHEMBL8532716 0.77 PIN1 (0.59) PIN1CA2CA7ALDH1A1CYP1A2
SCHEMBL6266326 0.72 PIN1 (1.00) PIN1CA2CA7CTSLCTSS
SCHEMBL27284050 0.70 ALDH1A1 (0.71) PIN1CA2CA7ALDH1A1CYP1A2
SCHEMBL18328366 0.70 CA2 (0.56) PIN1CA2CA7ALDH1A1CYP1A2
SCHEMBL9765289 0.69 NR3C1 (0.62) PIN1CA2CA7CTSLCTSS
SCHEMBL21808621 0.69 CA2 (0.73) PIN1CA2CA7ALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6602883-B1 Inhibitors of farnesyl protein transferase BRISTOL-MYERS SQUIBB COMPANY 2003-08-05 US disclosed
US-6387926-B1 ANTICANCER AGENTS BRISTOL-MYERS SQUIBB COMPANY 2002-05-14 US disclosed