SCHEMBL7246633

SCHEMBL7246633

O=S(=O)(NC(CCBr)Cc1ccccc1)c1ccccc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 1/20 0.57
CA2 P00918 2/20 0.55
CA7 P43166 2/20 0.55
CTSL P07711 1/20 0.52
CTSS P25774 1/20 0.52
ALDH1A1 P00352 2/20 0.51
CYP1A2 P05177 1/20 0.51
CYP2C9 P11712 1/20 0.51
CYP2C19 P33261 1/20 0.51
MMP2 P08253 9/20 0.48
MMP9 P14780 6/20 0.48
ADAMTS4 O75173 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.46
CA1 P00915 1/20 0.46
CA4 P22748 1/20 0.46
CA9 Q16790 1/20 0.46
MMP1 P03956 1/20 0.46
MMP3 P08254 1/20 0.46
MMP7 P09237 1/20 0.46
MMP13 P45452 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7246631 1.00 PIN1 (0.57) PIN1CA2CA7CTSLCTSS
SCHEMBL8532716 0.81 PIN1 (0.59) PIN1CA2CA7CTSLCTSS
Bromide SCHEMBL7245256 0.81 PIN1 (0.56) PIN1CA2CA7CTSLCTSS
Bromide SCHEMBL7245264 0.81 PIN1 (0.56) PIN1CA2CA7CTSLCTSS
SCHEMBL18328366 0.76 CA2 (0.56) PIN1CA2CA7CTSLCTSS
SCHEMBL3192784 0.75 CTSL (0.65) PIN1CA2CA7CTSLCTSS
SCHEMBL9298870 0.74 PIN1 (0.55) PIN1CA2CA7CTSLCTSS
SCHEMBL6266326 0.73 PIN1 (1.00) PIN1CA2CA7CTSLCTSS
SCHEMBL1287449 0.72 MMP2 (0.62) PIN1CA2CA7CTSLCTSS
SCHEMBL21808621 0.72 CA2 (0.73) PIN1CA2CA7CTSLCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6602883-B1 Inhibitors of farnesyl protein transferase BRISTOL-MYERS SQUIBB COMPANY 2003-08-05 US disclosed
US-6387926-B1 ANTICANCER AGENTS BRISTOL-MYERS SQUIBB COMPANY 2002-05-14 US disclosed