SCHEMBL7265407

SCHEMBL7265407

O=C[C@@H]1CCCN1C(=O)CCC(=O)NCc1cccc2ccccc12

nearest known ligand 0.64

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 1/20 0.53
PREP P48147 1/20 0.51
P2RX7 Q99572 1/20 0.48
MC4R P32245 2/20 0.44
MC1R Q01726 2/20 0.44
MC3R P41968 1/20 0.44
TSHR P16473 1/20 0.44
HDAC1 Q13547 1/20 0.43
HDAC8 Q9BY41 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
GAA P10253 1/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
PKM P14618 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7266965 0.85 PKM (0.55) SMN1; SMN2MEN1KMT2APKM
SCHEMBL7275011 0.85 NPC1 (0.54) PKM
SCHEMBL7266943 0.84 DPP4 (0.56) DPP4GAAMEN1KMT2A
SCHEMBL7275293 0.83 LMNA (0.45) DPP4PREPGAA
SCHEMBL7284471 0.83 DPP4 (0.47) DPP4PREPTSHRHDAC1HDAC8
SCHEMBL7272118 0.82 KDM4E (0.52) GAAMEN1KMT2APKM
SCHEMBL7316783 0.82 P2RX7 (0.43) DPP4PREPP2RX7HDAC1HDAC8
SCHEMBL7265335 0.80 P2RX7 (0.50) DPP4PREPP2RX7MC4RMC1R
SCHEMBL7265331 0.79 KMT2A (0.46) DPP4PREPMEN1KMT2A
SCHEMBL7267106 0.79 TP53 (0.59) DPP4P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5340832-A Prolinal derivatives useful for treating amnesia ONO PHARMACEUTICAL CO., LTD. (JP) 1994-08-23 US claimed
EP-0268190-B1 PROLINAL DERIVATIVES ONO PHARMACEUTICAL CO., LTD. (JP) 1993-06-16 EP claimed
EP-0268190-A1 Prolinal derivatives ONO PHARMACEUTICAL CO., LTD. (JP) 1988-05-25 EP claimed
US-5340832-A Prolinal derivatives useful for treating amnesia ONO PHARMACEUTICAL CO., LTD. (JP) 1994-08-23 US disclosed
US-5254550-A Enzyme inhibitor ONO PHARMACEUTICAL CO., LTD. (JP) 1993-10-19 US disclosed
US-5100904-A Inhibition of prolyl endopeptidase ONO PHARMACEUTICAL CO., LTD. (JP) 1992-03-31 US disclosed