SCHEMBL7265665

SCHEMBL7265665

COC(=O)OC1=C(C)NC(C)=C(c2nc(C)no2)C1c1ccccc1[N+](=O)[O-]

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.51
KMT2A Q03164 6/20 0.51
ADORA3 P0DMS8 4/20 0.51
LMNA P02545 3/20 0.51
CYP1A2 P05177 3/20 0.51
CACNA1C Q13936 3/20 0.51
TP53 P04637 3/20 0.51
ABCC4 O15439 2/20 0.51
CACNA1F O60840 2/20 0.51
ABCB11 O95342 2/20 0.51
ADORA2A P29274 2/20 0.51
ADORA1 P30542 2/20 0.51
OPRM1 P35372 2/20 0.51
SCN1A P35498 2/20 0.51
HTR2B P41595 2/20 0.51
CACNA1D Q01668 2/20 0.51
KCNH2 Q12809 2/20 0.51
CACNA1S Q13698 2/20 0.51
SCN5A Q14524 2/20 0.51
SCN2A Q99250 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7273125 0.91 LMNA (0.47) MAPTKMT2AADORA3LMNACYP1A2
SCHEMBL7272935 0.87 ADORA3 (0.46) MAPTKMT2AADORA3LMNACYP1A2
SCHEMBL10997036 0.86 MAPT (0.68) MAPTKMT2AADORA3LMNACYP1A2
SCHEMBL7265676 0.85 ALDH1A1 (0.38) MAPTKMT2AADORA3LMNACYP1A2
SCHEMBL6427770 0.83 ADORA3 (0.67) MAPTKMT2AADORA3LMNACYP1A2
SCHEMBL10369519 0.83 ADORA3 (0.58) MAPTKMT2AADORA3LMNACYP1A2
SCHEMBL7264444 0.83 KMT2A (0.42) MAPTKMT2AADORA3CACNA1CTP53
SCHEMBL7263816 0.82 CYP2C9 (0.45) MAPTKMT2AADORA3LMNACYP1A2
SCHEMBL7264423 0.82 MEN1 (0.48) MAPTKMT2AADORA3LMNACYP1A2
SCHEMBL10998379 0.80 CACNA1C (0.54) MAPTKMT2AADORA3LMNACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0116708-A1 Substituted 1,4-dihydropyridines, method for their preparation and their use as pharmaceuticals CASSELLA Aktiengesellschaft (DE) 1984-08-29 EP disclosed