SCHEMBL7265773

SCHEMBL7265773

O=C(O)CN1CCNCCN(CC(=O)O)C(COCc2ccccc2)CN(CC(=O)O)CC1

nearest known ligand 0.45

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.45
SIGMAR1 Q99720 2/20 0.38
ALDH1A1 P00352 1/20 0.36
TACR1 P25103 1/20 0.36
KMT2A Q03164 1/20 0.36
CTSL P07711 1/20 0.35
CTSB P07858 1/20 0.35
CTSK P43235 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8478967 0.91 TACR1 (0.40) ALDH1A1TACR1CTSLCTSBCTSK
SCHEMBL3834075 0.83 SIGMAR1 (0.47) SIGMAR1ALDH1A1
SCHEMBL5547411 0.80 GLA (0.41) EGFRSIGMAR1ALDH1A1KMT2A
SCHEMBL3916786 0.80 AGTR2 (0.43) CTSLCTSBCTSK
SCHEMBL9024007 0.78 NR1D1 (0.39) KMT2A
SCHEMBL7264621 0.77 SIGMAR1 (0.37) SIGMAR1
SCHEMBL5547419 0.77 EGFR (0.41) EGFRSIGMAR1ALDH1A1KMT2A
SCHEMBL8478663 0.76 EGFR (0.49) EGFRALDH1A1KMT2A
SCHEMBL5800349 0.76 SIGMAR1 (0.38) SIGMAR1
SCHEMBL20997586 0.76 FOLH1 (0.40) EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE38329-E1 Chelated complexes of paramagnetic metals with low toxicity BRACCO IMAGING S.P.A. (IT) 2003-11-25 US disclosed
US-6177562-B1 Chelated complexes of paramagnetic metals with low toxicity DIBRA S.P.A. (IT) 2001-01-23 US disclosed