SCHEMBL9024007

SCHEMBL9024007

O=C(O)CN1CCN(CC(=O)O)CC(COCc2ccccc2)N(CC(=O)O)Cc2cccc(n2)C1

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NR1D1 P20393 1/20 0.39
ABHD6 Q9BV23 3/20 0.35
DAGLA Q9Y4D2 3/20 0.35
MEN1 O00255 1/20 0.35
GAA P10253 1/20 0.35
KMT2A Q03164 1/20 0.35
ACE P12821 1/20 0.35
GRM5 P41594 1/20 0.34
TEAD3 Q99594 1/20 0.33
AGTR2 P50052 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8478967 0.84 TACR1 (0.40) NR1D1TEAD3AGTR2
SCHEMBL9024977 0.82 SIGMAR1 (0.35)
SCHEMBL18807567 0.78 FOLH1 (0.34)
SCHEMBL16644695 0.78 CHIT1 (0.37)
SCHEMBL18807569 0.78 L3MBTL1 (0.38) MEN1KMT2A
SCHEMBL9906195 0.78 CHIT1 (0.37)
SCHEMBL10060134 0.78 CHIT1 (0.37)
SCHEMBL19389406 0.78 L3MBTL1 (0.38) MEN1KMT2A
SCHEMBL3834075 0.78 SIGMAR1 (0.47) AGTR2
SCHEMBL7265773 0.78 EGFR (0.45) KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0438206-B1 6-Ring-containing macrocyclic tetraaza compounds, processes for their preparation, and pharmaceutical agents containing them SCHERING AG (DE) 1996-08-21 EP disclosed
US-5403572-A Macrocyclic polyaza compounds containing 5 or 6 membered rings, process for producing them and pharmaceutical media containing them SCHERING AKTIENGESELLSCHAFT (DE) 1995-04-04 US disclosed
US-5334371-A Marcocyclic polyaza bicyclo compounds containing 5 or 6 membered rings, and method for MRI SCHERING AKTIENGESELLSCHAFT (DE) 1994-08-02 US disclosed
EP-0438206-A1 6-Ring-containing macrocyclic tetraaza compounds, processes for their preparation, and pharmaceutical agents containing them SCHERING AKTIENGESELLSCHAFT (DE) 1991-07-24 EP disclosed