SCHEMBL8478967

SCHEMBL8478967

O=C(O)CN1CCN(CC(=O)O)CCN(CC(=O)O)C(COCc2ccccc2)CN(CC(=O)O)CC1

nearest known ligand 0.42

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 1/20 0.40
SLC6A9 P48067 1/20 0.39
CTSL P07711 1/20 0.39
CTSB P07858 1/20 0.39
CTSK P43235 1/20 0.39
TEAD3 Q99594 1/20 0.39
AGTR2 P50052 1/20 0.38
NR1D1 P20393 1/20 0.38
ALDH1A1 P00352 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3834075 0.91 SIGMAR1 (0.47) AGTR2ALDH1A1
SCHEMBL7265773 0.91 EGFR (0.45) TACR1CTSLCTSBCTSKALDH1A1
SCHEMBL3916786 0.85 AGTR2 (0.43) SLC6A9CTSLCTSBCTSKAGTR2
SCHEMBL9024007 0.84 NR1D1 (0.39) TEAD3AGTR2NR1D1
SCHEMBL6858941 0.83 FOLH1 (0.44)
SCHEMBL3000798 0.83 FOLH1 (0.44)
SCHEMBL13567995 0.78 L3MBTL1 (0.46) ALDH1A1
SCHEMBL7573297 0.78 SIGMAR1 (0.56) ALDH1A1
SCHEMBL19590904 0.77 DPP4 (0.43)
SCHEMBL9032439 0.75 FOLH1 (0.45) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5922862-A Process for the preparation of tetraazamacrocycles DIBRA S.P.A. (IT) 1999-07-13 US claimed
US-5922862-A Process for the preparation of tetraazamacrocycles DIBRA S.P.A. (IT) 1999-07-13 US disclosed