SCHEMBL7270481

SCHEMBL7270481

CC(C)COC(=O)NC(CC[S+]([O-])CCC(NC(=O)OCC(C)C)c1ccccc1)c1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GPR88 Q9GZN0 2/20 0.41
ALDH1A1 P00352 4/20 0.40
TSHR P16473 4/20 0.40
LMNA P02545 3/20 0.40
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
POLB P06746 1/20 0.38
CTDSP1 Q9GZU7 1/20 0.38
KDM4E B2RXH2 1/20 0.38
HTT P42858 2/20 0.37
ALOX15 P16050 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
HPGD P15428 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7279578 0.82 MAPT (0.46) GPR88ALDH1A1TSHRLMNAPOLB
SCHEMBL7279722 0.81 GPR88 (0.42) GPR88ALDH1A1TSHRLMNAPOLB
SCHEMBL1890430 0.76 ALDH1A1 (0.50) ALDH1A1TSHRLMNAKDM4EHTT
SCHEMBL6436027 0.74 ATM (0.59) ALDH1A1TSHRLMNACYP1A2CYP3A4
SCHEMBL6436022 0.74 ATM (0.59) ALDH1A1TSHRLMNACYP1A2CYP3A4
SCHEMBL29858123 0.70 CYP1A2 (0.45) ALDH1A1CYP1A2KDM4E
SCHEMBL28824792 0.70 CYP1A2 (0.45) ALDH1A1CYP1A2KDM4E
SCHEMBL6923888 0.69 CTSK (0.55) LMNA
SCHEMBL1463820 0.68 ALDH1A1 (0.49) ALDH1A1TSHRLMNACYP1A2CYP3A4
SCHEMBL14654947 0.68 NPC1 (0.63) ALDH1A1TSHRLMNAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0839798-A2 Intermediates for preparating non-peptide retroviral protease inhibitors ABBOTT LABORATORIES (US) 1998-05-06 EP disclosed
US-5670675-A Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1997-09-23 US disclosed
US-5545750-A TREATING HUMAN IMMUNODEFICIENCY VIRUS ABBOTT LABORATORIES (US) 1996-08-13 US disclosed
US-5142056-A Human immunodeficiency virus protease inhibitor ABBOTT LABORATORIES (US) 1992-08-25 US disclosed
EP-0402646-A1 Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1990-12-19 EP disclosed