SCHEMBL7279722

SCHEMBL7279722

CC(C)COC(=O)NC(CCS(=O)(=O)CCC(NC(=O)OCC(C)C)c1ccccc1)c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GPR88 Q9GZN0 1/20 0.42
KCNA5 P22460 1/20 0.41
ALDH1A1 P00352 3/20 0.41
TSHR P16473 2/20 0.41
LMNA P02545 3/20 0.41
POLB P06746 1/20 0.39
CTDSP1 Q9GZU7 1/20 0.39
KDM4E B2RXH2 1/20 0.39
RAB9A P51151 1/20 0.39
CCR5 P51681 1/20 0.38
HTT P42858 2/20 0.38
ALOX15 P16050 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7279578 0.83 MAPT (0.46) GPR88ALDH1A1TSHRLMNAPOLB
SCHEMBL7270481 0.81 GPR88 (0.41) GPR88ALDH1A1TSHRLMNAPOLB
SCHEMBL1890430 0.77 ALDH1A1 (0.50) ALDH1A1TSHRLMNAKDM4EHTT
SCHEMBL6436022 0.75 ATM (0.59) ALDH1A1TSHRLMNAKDM4ERAB9A
SCHEMBL6436027 0.75 ATM (0.59) ALDH1A1TSHRLMNAKDM4ERAB9A
SCHEMBL7407225 0.72 MMP13 (0.48) ALDH1A1TSHRLMNA
SCHEMBL12482203 0.71 ROCK1 (0.51) GPR88ALDH1A1TSHRLMNA
SCHEMBL28911342 0.71 CTSK (0.49) ALDH1A1TSHRLMNARAB9AHTT
SCHEMBL28911341 0.71 CTSK (0.49) ALDH1A1TSHRLMNARAB9AHTT
SCHEMBL29858123 0.71 CYP1A2 (0.45) ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0839798-A2 Intermediates for preparating non-peptide retroviral protease inhibitors ABBOTT LABORATORIES (US) 1998-05-06 EP disclosed
US-5670675-A Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1997-09-23 US disclosed
US-5142056-A Human immunodeficiency virus protease inhibitor ABBOTT LABORATORIES (US) 1992-08-25 US disclosed
EP-0402646-A1 Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1990-12-19 EP disclosed