SCHEMBL7273443

SCHEMBL7273443

Nc1cccc(-c2cccc(C(=O)NC[C@@H]3C[C@@H](CC(=O)O)C(=O)N3CCCc3ccccc3)c2)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.42
CFD P00746 1/20 0.38
CHRM3 P20309 1/20 0.38
DRD2 P14416 2/20 0.37
DRD4 P21917 1/20 0.37
KDM4B O94953 1/20 0.36
SMYD2 Q9NRG4 1/20 0.36
SENP1 Q9P0U3 1/20 0.36
ALDH1A1 P00352 1/20 0.36
TSHR P16473 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
OPRM1 P35372 1/20 0.35
OPRD1 P41143 1/20 0.35
OPRK1 P41145 1/20 0.35
KCNH2 Q12809 1/20 0.35
SIGMAR1 Q99720 1/20 0.35
HDAC1 Q13547 1/20 0.35
ERN1 O75460 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7283245 0.94 DRD2 (0.43) HTR1ADRD2DRD4ALDH1A1TSHR
SCHEMBL7275712 0.92 HTR1A (0.41) HTR1ACFDCHRM3DRD2SENP1
SCHEMBL7284946 0.89 F10 (0.48) HTR1A
SCHEMBL7275519 0.88 HTR1A (0.44) HTR1ACFDDRD2ALDH1A1TSHR
SCHEMBL7274585 0.87 ITGB3 (0.42) HTR1ASENP1
SCHEMBL7283567 0.87 DRD2 (0.44) HTR1ADRD2DRD4ALDH1A1TSHR
SCHEMBL7275596 0.86 DRD2 (0.41) HTR1ADRD2DRD4OPRM1OPRD1
SCHEMBL7274776 0.86 ITGB3 (0.45) HTR1AOPRM1OPRD1
Methyl Alcohol SCHEMBL8879759 0.86 HTR1A (0.40) HTR1ACHRM3DRD2
Hydrochloric Acid SCHEMBL7272974 0.86 F10 (0.51)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0483667-B1 Cyclic imino derivatives, process for their preparation and drugs containing them THOMAE GMBH DR K (DE) 1998-02-04 EP disclosed
US-5591769-A PYRROLIDINE DERIVATIVES; ANTICOAGULANTS KARL THOMAE GMBH (DE) 1997-01-07 US disclosed
US-5541343-A ANTIAGGLOMERANTS FOR CELLS OR ANTICOAGULANTS KARL THOMAE GMBH (DE) 1996-07-30 US disclosed
EP-0483667-A2 Cyclic imino derivatives, process for their preparation and drugs containing them Dr. Karl Thomae GmbH (DE) 1992-05-06 EP disclosed