SCHEMBL7275596

SCHEMBL7275596

COC(=O)C[C@@H]1C[C@@H](CNC(=O)c2ccc(-c3cccc(N)c3)cc2)N(CCCc2ccccc2)C1=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.41
DRD4 P21917 1/20 0.41
F10 P00742 1/20 0.38
OPRM1 P35372 2/20 0.38
OPRD1 P41143 2/20 0.38
LMNA P02545 1/20 0.38
HTR1A P08908 2/20 0.37
EGFR P00533 1/20 0.36
DRD3 P35462 1/20 0.36
PTAFR P25105 1/20 0.36
SLC6A2 P23975 1/20 0.35
SLC6A4 P31645 1/20 0.35
CHRNB2 P17787 1/20 0.35
CHRNB4 P30926 1/20 0.35
CHRNA3 P32297 1/20 0.35
CHRNA4 P43681 1/20 0.35
HDAC1 Q13547 3/20 0.35
ITGB3 P05106 1/20 0.35
ITGA2B P08514 1/20 0.35
HDAC3 O15379 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7275712 0.94 HTR1A (0.41) DRD2OPRM1OPRD1HTR1ADRD3
SCHEMBL7273413 0.92 DRD2 (0.42) DRD2DRD4F10OPRM1OPRD1
SCHEMBL7283245 0.92 DRD2 (0.43) DRD2DRD4F10HTR1AEGFR
Hydrochloric Acid SCHEMBL7275887 0.89 F10 (0.49) F10HTR1A
SCHEMBL7273369 0.89 MAOA (0.38) DRD2HTR1ADRD3
SCHEMBL7284968 0.88 ALDH1A1 (0.43) HDAC2
Hydrochloric Acid SCHEMBL7272455 0.88 F10 (0.45) F10HTR1AITGB3ITGA2B
Hydrochloric Acid SCHEMBL7279790 0.87 F10 (0.42) F10OPRM1OPRD1LMNAITGB3
SCHEMBL7273443 0.86 HTR1A (0.42) DRD2DRD4OPRM1OPRD1HTR1A
SCHEMBL7274708 0.86 CHRM4 (0.42) DRD4OPRM1OPRD1LMNAHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0483667-B1 Cyclic imino derivatives, process for their preparation and drugs containing them THOMAE GMBH DR K (DE) 1998-02-04 EP disclosed
US-5591769-A PYRROLIDINE DERIVATIVES; ANTICOAGULANTS KARL THOMAE GMBH (DE) 1997-01-07 US disclosed
US-5541343-A ANTIAGGLOMERANTS FOR CELLS OR ANTICOAGULANTS KARL THOMAE GMBH (DE) 1996-07-30 US disclosed
EP-0483667-A2 Cyclic imino derivatives, process for their preparation and drugs containing them Dr. Karl Thomae GmbH (DE) 1992-05-06 EP disclosed