SCHEMBL7284968

SCHEMBL7284968

COC(=O)C[C@@H]1C[C@@H](CNC(=O)c2ccc(-c3cccc([N+](=O)[O-])c3)cc2)N(CCCc2ccccc2)C1=O

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.43
HPGD P15428 2/20 0.43
P2RX7 Q99572 4/20 0.41
RAB9A P51151 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.40
SIGMAR1 Q99720 2/20 0.40
MAPT P10636 1/20 0.39
NPC1 O15118 1/20 0.38
TAAR1 Q96RJ0 1/20 0.38
PKM P14618 1/20 0.38
PLG P00747 1/20 0.37
PLAU P00749 1/20 0.37
PLAT P00750 1/20 0.37
HDAC2 Q92769 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7280821 0.95 ALDH1A1 (0.47) ALDH1A1HPGDRAB9ASMN1; SMN2SIGMAR1
SCHEMBL7275560 0.93 ALDH1A1 (0.45) ALDH1A1HPGDP2RX7RAB9ASMN1; SMN2
SCHEMBL7275596 0.88 DRD2 (0.41) HDAC2
SCHEMBL7273369 0.86 MAOA (0.38) RAB9AMAPT
Hydrochloric Acid SCHEMBL7275887 0.85 F10 (0.49) PLG
Hydrochloric Acid SCHEMBL7272455 0.84 F10 (0.45) PLG
SCHEMBL7274708 0.83 CHRM4 (0.42) HPGDRAB9ASIGMAR1
Hydrochloric Acid SCHEMBL7279790 0.83 F10 (0.42)
SCHEMBL7273655 0.83 SIGMAR1 (0.40) ALDH1A1HPGDRAB9ASMN1; SMN2SIGMAR1
SCHEMBL7278834 0.83 HTR1A (0.39) HPGDRAB9APLAU

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0483667-B1 Cyclic imino derivatives, process for their preparation and drugs containing them THOMAE GMBH DR K (DE) 1998-02-04 EP disclosed
US-5591769-A PYRROLIDINE DERIVATIVES; ANTICOAGULANTS KARL THOMAE GMBH (DE) 1997-01-07 US disclosed
US-5541343-A ANTIAGGLOMERANTS FOR CELLS OR ANTICOAGULANTS KARL THOMAE GMBH (DE) 1996-07-30 US disclosed
EP-0483667-A2 Cyclic imino derivatives, process for their preparation and drugs containing them Dr. Karl Thomae GmbH (DE) 1992-05-06 EP disclosed