SCHEMBL7277331

SCHEMBL7277331

CC1(C)C=C(n2ccccc2=O)c2cc(C(N)=O)ccc2O1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F10 P00742 5/20 0.40
KDM4E B2RXH2 1/20 0.34
BRD4 O60885 1/20 0.34
ALDH1A1 P00352 1/20 0.34
BRPF1 P55201 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
HSD17B10 Q99714 1/20 0.34
RARA P10276 1/20 0.34
RARB P10826 1/20 0.34
RARG P13631 1/20 0.34
BAZ2B Q9UIF8 1/20 0.33
BAZ2A Q9UIF9 1/20 0.33
PDK2 Q15119 1/20 0.33
TSHR P16473 1/20 0.33
CYP2D6 P10635 1/20 0.32
OPRM1 P35372 1/20 0.32
OPRD1 P41143 1/20 0.32
OPRK1 P41145 1/20 0.32
KCNH2 Q12809 1/20 0.32
AKT1 P31749 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8085330 0.91 F10 (0.40) F10KDM4EBRD4ALDH1A1BRPF1
SCHEMBL7276973 0.90 F10 (0.33) F10RARARARBRARG
SCHEMBL8090551 0.90 RARA (0.41) KDM4EALDH1A1HSD17B10RARARARB
SCHEMBL7277136 0.90 S100A4 (0.38) F10KDM4EALDH1A1RARARARB
SCHEMBL7268034 0.87 ALOX5 (0.40) F10ALDH1A1SMN1; SMN2RARARARB
SCHEMBL8088448 0.86 RARA (0.32) F10RARARARBRARG
SCHEMBL8088450 0.86 RARA (0.32) RARARARBRARG
SCHEMBL10696935 0.85 MAPT (0.34) KDM4EBRD4ALDH1A1BRPF1SMN1; SMN2
SCHEMBL9735586 0.84 F10 (0.39) F10KDM4EBRD4ALDH1A1BRPF1
SCHEMBL7277024 0.84 ALDH1A1 (0.42) KDM4EALDH1A1SMN1; SMN2HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6153627-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-11-28 US disclosed
US-6040308-A Chroman derivatives MERCK GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-03-21 US disclosed
US-5387587-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1995-02-07 US disclosed
EP-0346724-A1 Chroman derivates MERCK PATENT GmbH (DE) 1989-12-20 EP disclosed
EP-0273262-A2 Chroman derivatives MERCK PATENT GmbH (DE) 1988-07-06 EP disclosed