SCHEMBL7277136

SCHEMBL7277136

CC(=O)c1ccc2c(c1)C(n1ccccc1=O)=CC(C)(C)O2

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
S100A4 P26447 1/20 0.38
KDM4E B2RXH2 3/20 0.34
RARA P10276 1/20 0.34
RARB P10826 1/20 0.34
RARG P13631 1/20 0.34
NR1H2 P55055 1/20 0.34
NR1H3 Q13133 1/20 0.34
F10 P00742 3/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
PDK2 Q15119 1/20 0.31
ITGB1 P05556 1/20 0.31
ITGA4 P13612 1/20 0.31
MEN1 O00255 1/20 0.30
ALDH1A1 P00352 1/20 0.30
KMT2A Q03164 1/20 0.30
FGFR1 P11362 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8090551 0.91 RARA (0.41) KDM4ERARARARBRARGNR1H2
SCHEMBL7277331 0.90 F10 (0.40) KDM4ERARARARBRARGF10
SCHEMBL8088448 0.90 RARA (0.32) RARARARBRARGF10
SCHEMBL7268034 0.88 ALOX5 (0.40) RARARARBRARGF10NPC1
SCHEMBL8088450 0.87 RARA (0.32) RARARARBRARG
SCHEMBL7276973 0.86 F10 (0.33) RARARARBRARGF10
SCHEMBL8085176 0.85 MAOA (0.42) F10NPC1RAB9APDK2MEN1
SCHEMBL8204761 0.85 S100A4 (0.36) S100A4KDM4ENR1H2NR1H3F10
SCHEMBL10697122 0.85 MAPT (0.34) S100A4KDM4ERARARARBRARG
SCHEMBL7277024 0.85 ALDH1A1 (0.42) KDM4ERAB9AMEN1ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6153627-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-11-28 US disclosed
US-5391751-A Hypotensive, antiarrhythmia, antiasthmatic agents RED BALLOON INVESTMENT LIMITED (JE) 1995-02-21 US disclosed
US-5387587-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1995-02-07 US disclosed
US-5043352-A Chroman derivatives for the treatment of depressive states SANOFI (FR) 1991-08-27 US disclosed
EP-0346724-A1 Chroman derivates MERCK PATENT GmbH (DE) 1989-12-20 EP disclosed
EP-0273262-A2 Chroman derivatives MERCK PATENT GmbH (DE) 1988-07-06 EP disclosed