SCHEMBL7281990

SCHEMBL7281990

CCOC(=O)C1=C(C)Nc2c(c(C)nn2C)C1c1ccccc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 1/20 0.58
KDM4E B2RXH2 7/20 0.52
ALDH1A1 P00352 6/20 0.52
GAA P10253 3/20 0.52
SMN1; SMN2 Q16637 2/20 0.52
TSHR P16473 1/20 0.52
ACHE P22303 1/20 0.51
HSD17B10 Q99714 2/20 0.48
CASP1 P29466 1/20 0.48
ABCC1 P33527 1/20 0.48
CACNA1D Q01668 2/20 0.47
CACNA1F O60840 1/20 0.47
CACNA1S Q13698 1/20 0.47
CACNA1C Q13936 1/20 0.47
DHFR P00374 1/20 0.47
LMNA P02545 1/20 0.47
HPGD P15428 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7273090 0.87 ACHE (0.54) ADORA3KDM4EALDH1A1SMN1; SMN2TSHR
SCHEMBL7282275 0.87 CA1 (0.49) ADORA3KDM4EALDH1A1GAASMN1; SMN2
SCHEMBL7273692 0.87 ACHE (0.56) ADORA3KDM4EALDH1A1GAATSHR
SCHEMBL7278639 0.85 TSHR (0.52) ADORA3KDM4EALDH1A1GAATSHR
SCHEMBL7278678 0.84 CACNA1F (0.70) ADORA3TSHRACHECACNA1DCACNA1F
SCHEMBL4261000 0.83 MAPT (0.56) ADORA3KDM4EALDH1A1GAASMN1; SMN2
SCHEMBL7282331 0.81 ACHE (0.56) ADORA3KDM4EALDH1A1SMN1; SMN2TSHR
SCHEMBL16747575 0.79 GAA (0.68) ADORA3KDM4EALDH1A1GAASMN1; SMN2
SCHEMBL7280226 0.79 ACHE (0.52) ADORA3KDM4EALDH1A1GAAACHE
SCHEMBL3027412 0.79 ADORA3 (0.89) ADORA3KDM4EALDH1A1GAASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0114273-B1 NEW PHARMACOLOGICALLY ACTIVE PYRAZOLOPYRIDINES GRUPPO LEPETIT S.p.A. (IT) 1991-11-06 EP disclosed
US-4954508-A HYPOTENSIVE GRUPPO LEPETIT S.P.A. (IT) 1990-09-04 US disclosed