SCHEMBL7283137

SCHEMBL7283137

CC(=O)C(C(=O)O)C(S)c1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.45
SRC P12931 1/20 0.45
PDPK1 O15530 2/20 0.44
LMNA P02545 4/20 0.43
MAPK1 P28482 2/20 0.43
TDP1 Q9NUW8 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
ALDH1A1 P00352 2/20 0.41
CYP3A4 P08684 2/20 0.41
HPGD P15428 2/20 0.40
MAPT P10636 2/20 0.40
PTGS1 P23219 2/20 0.40
CXCR1 P25024 2/20 0.40
CXCR2 P25025 2/20 0.40
PTGS2 P35354 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
RECQL P46063 1/20 0.40
KDM4E B2RXH2 1/20 0.40
PMP22 Q01453 1/20 0.40
SLC22A6 Q4U2R8 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11390783 0.79 BRD4 (0.53) CYP2D6SRCLMNAMAPK1ALDH1A1
SCHEMBL9671856 0.78 CYP2D6 (0.46) CYP2D6SRCLMNAMAPK1ALDH1A1
SCHEMBL6159580 0.78 CYP2D6 (0.46) CYP2D6SRCLMNAMAPK1ALDH1A1
SCHEMBL5880392 0.77 HKDC1 (0.47) CYP2D6SRCPDPK1LMNAMAPK1
SCHEMBL28787458 0.76 DPP4 (0.50) CYP2D6SRCLMNAMAPK1PTGS1
SCHEMBL23743139 0.75 CYP2D6 (0.48) CYP2D6SRCLMNAMAPK1TDP1
SCHEMBL7434255 0.74 ALPI (0.50) CYP2D6PDPK1TDP1L3MBTL1MAPT
SCHEMBL6691791 0.74 BRD4 (0.63) CYP2D6SRCLMNAMAPK1TDP1
SCHEMBL7343000 0.74 CYP2D6 (0.46) CYP2D6SRCLMNAMAPK1TDP1
SCHEMBL8925590 0.72 LMNA (0.54) CYP2D6SRCLMNAMAPK1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5786494-A Process for the synthesis of α-substituted acrylic acids and their application SOCIETE CIVILE BIOPROJET (FR) 1998-07-28 US disclosed
EP-0481522-A1 Novel mercaptoacetylamide derivatives useful as inhibitors of enkephalinase and ace MERRELL PHARMACEUTICALS INC. (US) 1992-04-22 EP disclosed