SCHEMBL728343

SCHEMBL728343

NC(=S)Nc1ccc(N)cc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.62
TP53 P04637 1/20 0.62
TYR P14679 1/20 0.62
TSHR P16473 1/20 0.62
TAS2R38 P59533 1/20 0.62
HSD17B10 Q99714 1/20 0.62
CYP3A4 P08684 1/20 0.61
CYP2D6 P10635 1/20 0.61
CYP2C9 P11712 1/20 0.61
HPGD P15428 1/20 0.61
ALOX12 P18054 1/20 0.61
CYP2C19 P33261 1/20 0.61
KMT2A Q03164 4/20 0.59
MAPT P10636 3/20 0.59
RAB9A P51151 2/20 0.59
MEN1 O00255 2/20 0.59
SMN1; SMN2 Q16637 2/20 0.57
GAA P10253 1/20 0.57
KIF11 P52732 1/20 0.52
LMNA P02545 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL725810 0.89 ALDH1A1 (0.75) ALDH1A1TP53TYRTSHRTAS2R38
SCHEMBL12070412 0.83 MAPT (0.69) ALDH1A1TAS2R38HSD17B10CYP3A4CYP2C9
SCHEMBL14872162 0.83 TAS2R38 (0.60) ALDH1A1TP53TYRTSHRTAS2R38
SCHEMBL1822006 0.80 ALDH1A1 (0.65) ALDH1A1TP53TYRTSHRTAS2R38
SCHEMBL12071790 0.80 ALDH1A1 (0.62) ALDH1A1TP53TYRTSHRTAS2R38
Ammonia Solution, Strong SCHEMBL11429312 0.79 MAPT (0.59) ALDH1A1TP53TYRTSHRTAS2R38
SCHEMBL5518697 0.78 IDO1 (0.63) ALDH1A1TP53TYRTSHRTAS2R38
SCHEMBL526059 0.78 MAPT (0.63) ALDH1A1TP53TYRTSHRTAS2R38
SCHEMBL449122 0.78 ALDH1A1 (0.60) ALDH1A1TP53TYRTSHRTAS2R38
SCHEMBL11751583 0.78 ALDH1A1 (0.61) ALDH1A1TP53TYRTSHRTAS2R38

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5236633-A Blend of transparent polymer, thiourea and copper compounds JUJO PAPER CO., LTD. (JP) 1993-08-17 US claimed
US-4264710-A AN ETHYLENICALLY UNSATURATED COMPOUND, AND A PHOTOPOLYMERIZATION INIATOR FUJI PHOTO FILM CO., LTD. (JP) 1981-04-28 US claimed
CN-114249702-B N-aryl- [2,4 '-dithiazole ] -2' -amine compound and preparation and application thereof 沈阳药科大学 2023-09-05 CN disclosed
CN-114249702-A N-aryl- [2,4 '-bithiazole ] -2' -amine compound and preparation and application thereof 沈阳药科大学 2022-03-29 CN disclosed
CN-113631663-A Sulfonated 2(7) -aminoacridone and 1-aminopyrene dyes and their use as fluorescent labels, in particular for carbohydrate analysis 马克斯·普朗克科学促进学会 2021-11-09 CN disclosed
WO-2011152471-A2 RECHARGEABLE BATTERY, FUNCTIONAL POLYMER, AND METHOD FOR SYNTHESIS THEREOF 株式会社ポリチオン (JP) 2011-12-08 WO disclosed
US-20100298340-A1 Thiazol-Guanidine Derivatives Useful As A (Beta)-Related Pathologies ASTRAZENECA AB (SE) 2010-11-25 US disclosed
CN-101466692-A Thiazol-guanidine derivatives useful as a (beta) - related pathologies ASTRAZENECA AB (SE) 2009-06-24 CN disclosed
EP-2010508-A1 THIAZOL-GUANIDINE DERIVATIVES USEFUL AS A (BETA)- RELATED PATHOLOGIES AstraZeneca AB (SE) 2009-01-07 EP disclosed
US-20080227895-A1 Fire retardant vinyl chloride-based resin composition and molded article thereof MITSUBISHI PLASTICS, INC. (JP) 2008-09-18 US disclosed
WO-2007120096-A1 THIAZOL-GUANIDINE DERIVATIVES USEFUL AS A (BETA)- RELATED PATHOLOGIES ASTRAZENECA AB (SE) 2007-10-25 WO disclosed
CN-1315936-C Flame-resistant vinyl chloride based resin composition and formed product therefrom MITSUBISHI PLASTICS INC (JP) 2007-05-16 CN disclosed
US-20060014874-A1 Flame-resistant vinyl chlorride based resin composition and formed product therefrom MITSUBISHI PLASTICS, INC. (JP) 2006-01-19 US disclosed
CN-1708550-A Flame-resistant vinyl chloride based resin composition and formed product therefrom MITSUBISHI PLASTICS INC (JP) 2005-12-14 CN disclosed
CN-1054803-C Polycarbonic acid ester resin layered products absorbing near-infrared and formed products made of same DAICEL CHEM (JP) 2000-07-26 CN disclosed
US-5514740-A SHEET OR FILM HAVING CUPRIC SULFIDE DISPERSED THEREIN DAICEL CHEMICAL INDUSTRIES, LTD. (JP) 1996-05-07 US disclosed
US-5393443-A Hard-coating, heat-absorbing composition and heat-shielding substance JUJO PAPER CO., LTD. (JP) 1995-02-28 US disclosed
CN-1094354-A Polycarbonate-based resin laminate of absorption near infrared ray and formed body thereof DAICEL CHEM (JP) 1994-11-02 CN disclosed
US-4252963-A CYCLIZATION OF PHENYLTHIOUREAS WITH THIONYL CHLORIDE HOECHST AKTIENGESELLSCHAFT (DE) 1981-02-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100298340-A1 Thiazol-Guanidine Derivatives Useful As A (Beta)-Related Pathologies GRN, MAPT, GUCY1B1 ALDH1A1 1302/4885TP53 1888/4885TYR 3166/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.