SCHEMBL7284284

SCHEMBL7284284

CSc1ccc(/C=C/CCC2(c3cccc([N+](=O)[O-])c3)C(C(=O)O)=C(C)N(C)C(C)=C2C(=O)O)cc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 2/20 0.37
KMT2A Q03164 3/20 0.36
PTPN1 P18031 1/20 0.36
PTPN12 Q05209 1/20 0.36
PTPN22 Q9Y2R2 1/20 0.36
NFE2L2 Q16236 2/20 0.35
HTT P42858 2/20 0.35
ALDH1A1 P00352 2/20 0.35
CDK2 P24941 1/20 0.35
MAPT P10636 3/20 0.35
GSK3B P49841 1/20 0.34
MEN1 O00255 2/20 0.34
MLNR O43193 1/20 0.34
NR1I2 O75469 1/20 0.34
CACNA1H O95180 1/20 0.34
NR3C1 P04150 1/20 0.34
ADORA3 P0DMS8 1/20 0.34
TBXA2R P21731 1/20 0.34
PDE4D Q08499 1/20 0.34
CACNA1C Q13936 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9831502 0.86 MAOB (0.40) CACNA1BKMT2ANFE2L2HTTALDH1A1
SCHEMBL7326485 0.82 CACNA1B (0.45) CACNA1BKMT2APTPN1PTPN12PTPN22
SCHEMBL9249991 0.82 CACNA1B (0.45) CACNA1BKMT2APTPN1PTPN12PTPN22
SCHEMBL7365756 0.81 CACNA1B (0.40) CACNA1BKMT2APTPN1PTPN12PTPN22
SCHEMBL8827906 0.78 ALDH1A1 (0.39) KMT2AALDH1A1MAPTKDM4ESMN1; SMN2
SCHEMBL7366816 0.78 CACNA1B (0.39) CACNA1BKMT2APTPN1PTPN12PTPN22
SCHEMBL4883866 0.77 TP53 (0.43) KMT2AALDH1A1MAPTMEN1ADORA3
SCHEMBL7275212 0.75 SIGMAR1 (0.45) KMT2AHTTALDH1A1CDK2MAPT
SCHEMBL7283842 0.74 MEN1 (0.38) CACNA1BKMT2ANFE2L2HTTALDH1A1
SCHEMBL7267935 0.74 LMNA (0.44) KMT2AALDH1A1MAPTMEN1ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0173126-A1 Process for preparing novel dihydropyridine derivatives OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1986-03-05 EP disclosed