SCHEMBL7289569

SCHEMBL7289569

CCC1(c2cccc(Cl)c2Cl)C(C(=O)O)=C(C)N(CCN2CCC(C(c3ccccc3)c3ccccc3)CC2)C(C)=C1C(=O)O

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 2/20 0.36
CCR5 P51681 1/20 0.35
TACR2 P21452 1/20 0.35
PRCP P42785 2/20 0.35
OPRM1 P35372 1/20 0.35
CHRM2 P08172 1/20 0.34
HTR1A P08908 1/20 0.34
CHRM1 P11229 1/20 0.34
DRD2 P14416 1/20 0.34
ADRA1D P25100 1/20 0.34
ADRA1A P35348 1/20 0.34
ADRA1B P35368 1/20 0.34
CARM1 Q86X55 1/20 0.34
PRMT6 Q96LA8 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4758577 0.77 TSHR (0.36) ADRA1A
SCHEMBL9101372 0.76 TSHR (0.37) DRD2ADRA1A
SCHEMBL4757355 0.70 PYGM (0.39)
SCHEMBL11210015 0.70 CACNA2D1 (0.46) OPRM1CHRM2CHRM1DRD2ADRA1A
SCHEMBL10847722 0.66 CYP2C9 (0.59) OPRM1HTR1ACHRM1DRD2ADRA1D
SCHEMBL12123733 0.66 PRCP (0.55) BACE1CCR5PRCPCHRM2HTR1A
SCHEMBL4758583 0.66 PYGL (0.38) HTR1AADRA1A
SCHEMBL14282941 0.65 PRCP (0.54) BACE1PRCPCARM1PRMT6
SCHEMBL2365028 0.65 TSHR (0.37) ADRA1A
SCHEMBL4695183 0.65 PRCP (0.52) BACE1CCR5PRCPCHRM2HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0138505-A2 Dihydropyridine derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1985-04-24 EP disclosed