SCHEMBL4758583

SCHEMBL4758583

CCN1C(C)=C(C(=O)O)C(CC)(c2c(Cl)cccc2Cl)C(C(=O)O)=C1C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PYGL P06737 6/20 0.38
PYGM P11217 6/20 0.38
NOTUM Q6P988 3/20 0.35
TSHR P16473 1/20 0.33
AKR1B1 P15121 1/20 0.33
KMT2A Q03164 3/20 0.32
MEN1 O00255 2/20 0.32
TDP1 Q9NUW8 1/20 0.32
ALDH1A1 P00352 4/20 0.32
LMNA P02545 2/20 0.32
KDM4E B2RXH2 1/20 0.32
USP2 O75604 1/20 0.32
MT-CO2 P00403 1/20 0.32
TTR P02766 1/20 0.32
PLA2G1B P04054 1/20 0.32
CYP1A2 P05177 1/20 0.32
PGR P06401 1/20 0.32
CYP3A4 P08684 1/20 0.32
HTR1A P08908 1/20 0.32
ADRA2A P08913 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4758577 0.87 TSHR (0.36) PYGLPYGMNOTUMTSHRKMT2A
SCHEMBL4757355 0.86 PYGM (0.39) PYGLPYGMNOTUMALDH1A1LMNA
SCHEMBL4758254 0.81 HCAR3 (0.39) NOTUMTSHRTDP1ALDH1A1LMNA
SCHEMBL4758299 0.81 LMNA (0.42) PYGLPYGMTSHRKMT2AMEN1
SCHEMBL4757333 0.80 OPRM1 (0.36) NOTUMTSHRAKR1B1KMT2AALDH1A1
SCHEMBL4758575 0.80 OPRM1 (0.39) NOTUMTSHR
SCHEMBL4758286 0.79 TSHR (0.36) NOTUMTSHRALDH1A1LMNACYP3A4
SCHEMBL4757320 0.79 HCAR2 (0.39) NOTUMTSHRALDH1A1LMNAKDM4E
SCHEMBL4757340 0.77 NOTUM (0.34) NOTUML3MBTL1
SCHEMBL4756162 0.76 TDP1 (0.40) NOTUMTSHRKMT2ATDP1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008006070-A2 COMPOUNDS AND COMBINATIONS THEREOF FOR INHIBITING BETA-AMYLOID PRODUCTION AND METHODS OF USE THEREOF ROSKAMP RESEARCH LLC (US) 2008-01-10 WO disclosed