SCHEMBL7290042

SCHEMBL7290042

CC(=O)CC(=O)OCCN1CCN(c2ccccc2C)CC1

nearest known ligand 0.53

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 5/20 0.48
ADRA1A P35348 3/20 0.48
FAAH O00519 3/20 0.48
ADRA1D P25100 2/20 0.48
ADRA1B P35368 2/20 0.48
LMNA P02545 1/20 0.47
MAPT P10636 1/20 0.47
DRD2 P14416 4/20 0.47
CNR1 P21554 2/20 0.47
ALDH1A1 P00352 1/20 0.47
TSHR P16473 1/20 0.47
KMT2A Q03164 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
HTR7 P34969 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10365727 0.88 ADORA2B (0.55) DRD3LMNADRD2ALDH1A1HTR7
SCHEMBL10365793 0.85 DRD2 (0.61) DRD3DRD2ALDH1A1KMT2A
SCHEMBL10366024 0.83 SIGMAR1 (0.56) DRD3DRD2ALDH1A1KMT2AHTR7
SCHEMBL10365769 0.82 DRD2 (0.61) DRD3DRD2
SCHEMBL22882677 0.79 MGAM (0.43) DRD3DRD2ALDH1A1TSHRKMT2A
SCHEMBL314201 0.79 ALDH1A1 (0.56) DRD3ADRA1AADRA1DADRA1BMAPT
SCHEMBL10364966 0.78 HTR1A (0.63) DRD3DRD2HTR7
SCHEMBL10365050 0.78 MAOB (0.56) LMNAMAPTALDH1A1KMT2AHTR7
SCHEMBL11634761 0.78 TMEM97 (0.55) DRD3ADRA1AFAAHADRA1DADRA1B
SCHEMBL10367299 0.77 ADRA1B (0.52) ADRA1AADRA1DADRA1BLMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0094159-B1 DIHYDROPYRIDINE DERIVATIVES, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1990-03-14 EP disclosed
US-4892875-A HYPOTENSIVE, RENAL VASODILATION TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1990-01-09 US disclosed
EP-0138505-A2 Dihydropyridine derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1985-04-24 EP disclosed
EP-0094159-A1 Dihydropyridine derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1983-11-16 EP disclosed