SCHEMBL7301246

SCHEMBL7301246

c1ccc(-c2nc3cnc4c(c3[nH]2)CCCC4)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.41
GAA P10253 1/20 0.41
RAB9A P51151 1/20 0.41
GABRA1 P14867 1/20 0.40
GABRG2 P18507 1/20 0.40
GABRB3 P28472 1/20 0.40
GABRA3 P34903 1/20 0.40
ADORA2B P29275 1/20 0.39
TNKS O95271 1/20 0.39
PARP1 P09874 1/20 0.39
TNKS2 Q9H2K2 1/20 0.39
PI4KA P42356 1/20 0.38
PI4K2B Q8TCG2 1/20 0.38
PI4K2A Q9BTU6 1/20 0.38
PI4KB Q9UBF8 1/20 0.38
KMT2A Q03164 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
XDH P47989 1/20 0.38
FGFR1 P11362 1/20 0.38
FGFR2 P21802 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7301214 0.81 TNKS2 (0.43) NPC1GAARAB9AADORA2BTNKS
SCHEMBL7297879 0.76 SPR (0.34) GABRA1GABRG2GABRB3GABRA3
SCHEMBL1423662 0.71 TNKS (0.56) NPC1GAARAB9ATNKSPARP1
SCHEMBL1490653 0.71 GABRA1 (0.34) NPC1RAB9AGABRA1GABRG2GABRB3
SCHEMBL1032502 0.70 TNKS2 (0.68) TNKSPARP1TNKS2KMT2AL3MBTL1
SCHEMBL6861541 0.68 KMT2A (0.57) NPC1GAARAB9ATNKSPARP1
SCHEMBL9070566 0.67 TNKS (0.63) TNKSPARP1TNKS2KMT2AL3MBTL1
SCHEMBL10768720 0.67 TNKS (0.43) NPC1GAARAB9AADORA2BTNKS
SCHEMBL25696459 0.67 MAPK1 (0.48) NPC1GAARAB9AADORA2BTNKS
SCHEMBL14153754 0.66 KMT2A (0.54) NPC1GAARAB9ATNKSPARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0556008-B1 Condensed imidazopyridine derivatives with psychotropic activity SHIONOGI & CO (JP) 1997-05-14 EP disclosed
US-5461062-A Psychotropic agent as antianxiety agent, anesthesia antagonistic agent SHIONOGI & CO., LTD. (JP) 1995-10-24 US disclosed
US-5378848-A Benzodiazepine agonist, psychotropic, antianxiety, cerebral function activator, anesthesia atagonist SHIONOGI & CO., LTD. (JP) 1995-01-03 US disclosed
EP-0556008-A1 Condensed imidazopyridine derivatives with psychotropic activity SHIONOGI & CO., LTD. (JP) 1993-08-18 EP disclosed