SCHEMBL7302606

SCHEMBL7302606

COc1ccc(S(=O)(=O)C(CC2CCCC2)C(C(=O)NO)C(C)C)cc1

nearest known ligand 0.56

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MMP1 P03956 12/20 0.56
MMP3 P08254 8/20 0.56
MMP2 P08253 8/20 0.56
MMP13 P45452 10/20 0.55
MMP9 P14780 8/20 0.50
MMP8 P22894 2/20 0.49
ADAM17 P78536 5/20 0.48
PDE4A P27815 2/20 0.48
PDE4B Q07343 2/20 0.48
PDE4C Q08493 2/20 0.48
PDE4D Q08499 2/20 0.48
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CA9 Q16790 1/20 0.43
ALDH1A1 P00352 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7309436 0.88 MMP1 (0.50) MMP1MMP3MMP2MMP13MMP9
SCHEMBL7298812 0.77 MMP1 (0.42) MMP1MMP3MMP2MMP13MMP9
SCHEMBL7307517 0.77 ADAM17 (0.43) MMP1MMP3MMP2MMP13MMP9
SCHEMBL7309053 0.76 MMP3 (0.78) MMP1MMP3MMP2MMP13MMP9
SCHEMBL14188829 0.73 MMP1 (0.56) MMP1MMP3MMP2MMP13MMP9
SCHEMBL7306444 0.73 MMP1 (0.65) MMP1MMP3MMP2MMP13MMP9
SCHEMBL6928607 0.72 MMP1 (1.00) MMP1MMP3MMP2MMP13MMP9
SCHEMBL6934594 0.71 MMP1 (0.73) MMP1MMP3MMP2MMP13MMP9
SCHEMBL6931861 0.70 MMP1 (0.52) MMP1MMP3MMP2MMP13MMP9
SCHEMBL8714771 0.69 MMP13 (0.73) MMP1MMP3MMP2MMP13MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0780386-B1 Matrix metalloprotease inhibitors HOFFMANN LA ROCHE (CH) 2002-10-02 EP disclosed
US-5932595-A ANTIARTHRITIC AGENT; MULTIPLE SCLEROSIS; OSTEOPOROSIS; RESPIRATORY SYSTEM DISORDERS; SKIN DISORDERS; ANTIULCER AGENT SYNTEX (U.S.A.) INC. (US) 1999-08-03 US disclosed
EP-0780386-A1 Matrix metalloprotease inhibitors F. HOFFMANN-LA ROCHE AG (CH) 1997-06-25 EP disclosed