SCHEMBL7303142

SCHEMBL7303142

CN(C)c1ccc(-n2c(N)nc3ccccc32)cc1-c1ccco1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 4/20 0.42
ADORA1 P30542 3/20 0.41
ADORA2B P29275 3/20 0.41
KDM4E B2RXH2 8/20 0.40
ALDH1A1 P00352 7/20 0.40
TSHR P16473 4/20 0.40
PKM P14618 2/20 0.40
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
MEN1 O00255 2/20 0.40
BLM P54132 2/20 0.40
KMT2A Q03164 2/20 0.40
POLB P06746 1/20 0.40
CASP1 P29466 1/20 0.40
CASP7 P55210 1/20 0.40
HTT P42858 1/20 0.40
HPGD P15428 5/20 0.39
HSD17B10 Q99714 2/20 0.39
TP53 P04637 1/20 0.39
ADORA3 P0DMS8 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7299551 0.85 KDM4E (0.46) ADORA2AADORA1ADORA2BKDM4EALDH1A1
SCHEMBL7305553 0.82 ADORA2A (0.44) ADORA2AADORA1ADORA2BKDM4EALDH1A1
SCHEMBL7295510 0.77 TAAR1 (0.46) ADORA2AADORA1ADORA2BKDM4EALDH1A1
SCHEMBL7306716 0.76 ADORA2A (0.45) ADORA2AADORA1ADORA2BKDM4EALDH1A1
Oxalic Acid SCHEMBL7304901 0.71 KDM4E (0.46) ADORA2AADORA1ADORA2BKDM4EALDH1A1
SCHEMBL7298295 0.71 TAAR1 (0.46) ADORA2AADORA1ADORA2BKDM4EALDH1A1
SCHEMBL15214855 0.69 L3MBTL1 (0.56) ADORA2AADORA1KDM4EALDH1A1PKM
SCHEMBL7167684 0.69 NOS2 (0.53) KDM4EALDH1A1NPC1RAB9AMEN1
SCHEMBL23652406 0.69 KDM4E (0.55) ADORA2AADORA1KDM4EALDH1A1PKM
SCHEMBL17689831 0.68 NOS2 (0.49) NPC1RAB9AMEN1KMT2APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0604353-B1 Benzimidazole compounds, their preparation and use NEUROSEARCH AS (DK) 1998-07-01 EP claimed
US-5441969-A Imidazole compounds, their preparation and use NEUROSEARCH A/S (DK) 1995-08-15 US claimed
EP-0604353-A1 Benzimidazole compounds, their preparation and use NEUROSEARCH A/S (DK) 1994-06-29 EP claimed
EP-0604353-B1 Benzimidazole compounds, their preparation and use NEUROSEARCH AS (DK) 1998-07-01 EP disclosed
US-5441969-A Imidazole compounds, their preparation and use NEUROSEARCH A/S (DK) 1995-08-15 US disclosed
EP-0604353-A1 Benzimidazole compounds, their preparation and use NEUROSEARCH A/S (DK) 1994-06-29 EP disclosed