SCHEMBL7305553

SCHEMBL7305553

COc1ccc(-n2c(N)nc3ccccc32)cc1-c1ccco1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 4/20 0.44
PIK3R1 P27986 1/20 0.42
PIK3CA P42336 1/20 0.42
ADORA1 P30542 2/20 0.42
MAPT P10636 4/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
RPS6KB1 P23443 2/20 0.41
KDM4E B2RXH2 2/20 0.41
LMNA P02545 2/20 0.41
TSHR P16473 2/20 0.41
ALDH1A1 P00352 1/20 0.41
ALOX15 P16050 1/20 0.41
HSD17B10 Q99714 1/20 0.41
NPC1 O15118 4/20 0.41
RAB9A P51151 3/20 0.41
TP53 P04637 2/20 0.41
MAPK10 P53779 1/20 0.41
ADORA2B P29275 1/20 0.41
PTGS1 P23219 1/20 0.41
PTGS2 P35354 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7299551 0.85 KDM4E (0.46) ADORA2AADORA1MAPTSMN1; SMN2RPS6KB1
SCHEMBL7303142 0.82 ADORA2A (0.42) ADORA2AADORA1MAPTSMN1; SMN2KDM4E
SCHEMBL7295510 0.77 TAAR1 (0.46) ADORA2AADORA1MAPTSMN1; SMN2KDM4E
SCHEMBL7306716 0.76 ADORA2A (0.45) ADORA2AADORA1MAPTSMN1; SMN2RPS6KB1
SCHEMBL31452291 0.73 KDM4E (0.48) MAPTSMN1; SMN2RPS6KB1KDM4ETSHR
SCHEMBL6438855 0.72 ALDH1A1 (0.63) MAPTSMN1; SMN2RPS6KB1KDM4ELMNA
Oxalic Acid SCHEMBL7304901 0.71 KDM4E (0.46) ADORA2AADORA1MAPTSMN1; SMN2KDM4E
SCHEMBL7305407 0.71 ADORA2A (0.49) ADORA2APIK3R1PIK3CAADORA1MAPT
SCHEMBL7295792 0.70 RPS6KB1 (0.38) MAPTRPS6KB1LMNATSHRALDH1A1
SCHEMBL15214855 0.69 L3MBTL1 (0.56) ADORA2AADORA1MAPTSMN1; SMN2RPS6KB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0604353-B1 Benzimidazole compounds, their preparation and use NEUROSEARCH AS (DK) 1998-07-01 EP claimed
US-5441969-A Imidazole compounds, their preparation and use NEUROSEARCH A/S (DK) 1995-08-15 US claimed
EP-0604353-A1 Benzimidazole compounds, their preparation and use NEUROSEARCH A/S (DK) 1994-06-29 EP claimed
EP-0604353-B1 Benzimidazole compounds, their preparation and use NEUROSEARCH AS (DK) 1998-07-01 EP disclosed
US-5441969-A Imidazole compounds, their preparation and use NEUROSEARCH A/S (DK) 1995-08-15 US disclosed
EP-0604353-A1 Benzimidazole compounds, their preparation and use NEUROSEARCH A/S (DK) 1994-06-29 EP disclosed