SCHEMBL7304175

SCHEMBL7304175

CC(C)(C)OC(=O)C[C@H](NC(=O)CCNC(=O)c1ccc(C(=N)N)cc1)C(=O)N[C@@H](Cc1ccc(OC(C)(C)C)cc1)C(=O)OC(C)(C)C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 6/20 0.43
ITGA2B P08514 6/20 0.43
ABCB1 P08183 1/20 0.40
ADCY6 O43306 1/20 0.38
ADCY3 O60266 1/20 0.38
ADCY9 O60503 1/20 0.38
ADCY5 O95622 1/20 0.38
ADCY8 P40145 1/20 0.38
GCGR P47871 1/20 0.38
ADCY7 P51828 1/20 0.38
ADCY2 Q08462 1/20 0.38
ADCY1 Q08828 1/20 0.38
ADCY4 Q8NFM4 1/20 0.38
MMP1 P03956 3/20 0.38
PRSS1 P07477 3/20 0.37
TMPRSS15 P98073 2/20 0.37
CCKBR P32239 1/20 0.37
PLG P00747 1/20 0.36
PRSS2 P07478 1/20 0.36
PRSS3 P35030 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7296817 0.91 MAPT (0.44) ITGB3ITGA2BMMP1PRSS1CCKBR
Iodide SCHEMBL9221941 0.90 CCKBR (0.43) ITGB3ITGA2BMMP1PRSS1CCKBR
SCHEMBL9224835 0.87 ABCB1 (0.42) ITGB3ITGA2BABCB1MMP1PRSS1
Iodide SCHEMBL9217545 0.84 CCKBR (0.42) ITGB3ITGA2BMMP1CCKBRTMPRSS11D
SCHEMBL7302254 0.83 TDP1 (0.46) MMP1CCKBR
SCHEMBL7298759 0.82 ITGB3 (0.40) ITGB3ITGA2BPRSS1TMPRSS11D
Iodide SCHEMBL9223883 0.82 CCKBR (0.43) ADCY6ADCY3ADCY9ADCY5ADCY8
SCHEMBL7336100 0.81 CTSL (0.49) ITGB3ITGA2BABCB1CCKBR
SCHEMBL9218412 0.79 ST14 (0.47) ITGB3ITGA2BMMP1PRSS1TMPRSS15
SCHEMBL7301659 0.79 CTSG (0.46) ABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0445796-B1 Derivatives of acetic acid containing peptide bonds HOFFMANN LA ROCHE (CH) 1998-06-17 EP disclosed
US-5430024-A Peptides bearing N-terminal amidino moieties and their use as inhibitors of platelet aggregation HOFFMANN-LA ROCHE INC. (US) 1995-07-04 US disclosed
US-5273982-A An amidinoaryleneamidoalkylpiperazinyleneacetic acid HOFFMANN-LA ROCHE INC. (US) 1993-12-28 US disclosed
EP-0445796-A2 Derivatives of acetic acid F. HOFFMANN-LA ROCHE AG (CH) 1991-09-11 EP disclosed