SCHEMBL7302254

SCHEMBL7302254

CC(C)(C)OC(=O)C[C@H](NC(=O)CCNC(=O)c1ccc(C(N)=S)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)OC(C)(C)C

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 5/20 0.46
MAPT P10636 4/20 0.46
CCKBR P32239 1/20 0.45
POLB P06746 2/20 0.43
REN P00797 2/20 0.42
ACE P12821 1/20 0.42
KLK5 Q9Y337 1/20 0.41
ROCK2 O75116 2/20 0.41
MMP1 P03956 1/20 0.41
MMP3 P08254 1/20 0.41
MMP9 P14780 1/20 0.41
PAX8 Q06710 1/20 0.40
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
GLA P06280 1/20 0.40
ATM Q13315 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7307169 0.92 CCKBR (0.44) TDP1MAPTCCKBRPOLBREN
SCHEMBL7296817 0.92 MAPT (0.44) TDP1MAPTCCKBRPOLBREN
Iodide SCHEMBL9221941 0.91 CCKBR (0.43) TDP1MAPTCCKBRPOLBREN
SCHEMBL7301659 0.88 CTSG (0.46) TDP1MAPT
SCHEMBL7307254 0.87 MMP1 (0.49) TDP1MAPTPOLBRENACE
Iodide SCHEMBL9223883 0.87 CCKBR (0.43) TDP1MAPTCCKBRPOLBACE
SCHEMBL8438729 0.83 MEN1 (0.47) TDP1MAPTPOLBRENKLK5
Iodide SCHEMBL9217545 0.83 CCKBR (0.42) TDP1MAPTCCKBRRENACE
SCHEMBL7304175 0.83 ITGB3 (0.43) CCKBRMMP1
SCHEMBL9223666 0.82 REN (0.49) TDP1MAPTRENKLK5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0445796-B1 Derivatives of acetic acid containing peptide bonds HOFFMANN LA ROCHE (CH) 1998-06-17 EP disclosed
EP-0445796-A2 Derivatives of acetic acid F. HOFFMANN-LA ROCHE AG (CH) 1991-09-11 EP disclosed