SCHEMBL7336100

SCHEMBL7336100

CC(C)(C)OC(=O)C[C@H](NC(=O)CCNC(=O)OCc1ccccc1)C(=O)N[C@@H](Cc1ccc(OC(C)(C)C)cc1)C(=O)OC(C)(C)C

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CTSL P07711 1/20 0.49
CTSK P43235 1/20 0.49
ABCB1 P08183 1/20 0.48
CCKBR P32239 1/20 0.45
ACE P12821 1/20 0.43
ITGB3 P05106 1/20 0.43
ITGA2B P08514 1/20 0.43
KLK5 Q9Y337 2/20 0.43
REN P00797 1/20 0.43
PSMB10 P40306 1/20 0.42
PSMB2 P49721 1/20 0.42
MAPT P10636 2/20 0.42
KLK7 P49862 1/20 0.42
HTT P42858 1/20 0.41
TDP1 Q9NUW8 2/20 0.41
PSMB5 P28074 1/20 0.41
PAX8 Q06710 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9223970 0.86 CTSK (0.56) CTSLCTSKABCB1ITGB3ITGA2B
SCHEMBL30136171 0.84 LMNA (0.50) CTSLCTSKABCB1ACEITGB3
SCHEMBL7304574 0.84 MAPT (0.52) CTSLCTSKCCKBRACEKLK5
SCHEMBL8441060 0.83 CTSL (0.55) CTSLCTSK
SCHEMBL7304605 0.83 HTT (0.46) CTSLCTSKITGB3ITGA2BKLK5
SCHEMBL22457264 0.81 CTSL (0.61) CTSLCTSKABCB1ITGB3ITGA2B
SCHEMBL30645054 0.81 CTSB (0.50) CTSLCTSKCCKBRACEREN
SCHEMBL7304175 0.81 ITGB3 (0.43) ABCB1CCKBRITGB3ITGA2B
SCHEMBL16770322 0.80 CTSL (0.56) CTSLCTSKABCB1ITGB3ITGA2B
SCHEMBL7305886 0.79 CTSS (0.45) CTSLCTSKABCB1CCKBRACE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0445796-B1 Derivatives of acetic acid containing peptide bonds HOFFMANN LA ROCHE (CH) 1998-06-17 EP disclosed
US-5430024-A Peptides bearing N-terminal amidino moieties and their use as inhibitors of platelet aggregation HOFFMANN-LA ROCHE INC. (US) 1995-07-04 US disclosed
US-5273982-A An amidinoaryleneamidoalkylpiperazinyleneacetic acid HOFFMANN-LA ROCHE INC. (US) 1993-12-28 US disclosed