SCHEMBL7304441

SCHEMBL7304441

C=CCc1ccccc1OCC(O)CNCCc1nc2ccc(C3=NNC(=O)CC3C)cc2[nH]1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 12/20 0.43
HTR1A P08908 5/20 0.43
PDE3B Q13370 2/20 0.42
PDE3A Q14432 2/20 0.42
ABCB11 O95342 1/20 0.42
MAOA P21397 1/20 0.42
ADORA2A P29274 1/20 0.42
TP53 P04637 1/20 0.42
MAPT P10636 1/20 0.42
ALDH1A1 P00352 1/20 0.41
F10 P00742 1/20 0.41
ADRB1 P08588 4/20 0.40
LMNA P02545 2/20 0.40
ADRB3 P13945 2/20 0.40
ADRA2C P18825 1/20 0.40
SLC6A2 P23975 1/20 0.40
BDKRB2 P30411 1/20 0.40
SLC6A4 P31645 1/20 0.40
ADRA1A P35348 1/20 0.40
HTR2B P41595 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7304427 0.95 ADRB2 (0.43) ADRB2HTR1ATP53MAPTALDH1A1
SCHEMBL7305060 0.92 PDE3B (0.43) ADRB2HTR1APDE3BPDE3AABCB11
SCHEMBL7305054 0.86 SLC22A1 (0.39) ADRB2HTR1APDE3BPDE3AABCB11
SCHEMBL7304010 0.86 PDE3B (0.43) ADRB2PDE3BPDE3AABCB11MAOA
SCHEMBL9687171 0.82 PDE3B (0.41) PDE3BPDE3AABCB11MAOAADORA2A
SCHEMBL9687447 0.82 MAPK1 (0.41) ADRB2HTR1APDE3BPDE3ATP53
SCHEMBL7297393 0.81 PDE3B (0.47) ADRB2PDE3BPDE3AABCB11MAOA
SCHEMBL7303996 0.81 CTSS (0.43) ADRB2ADRB1ADRB3CYP1A2KDM4E
SCHEMBL7304432 0.79 ALDH1A1 (0.45) ADRB2HTR1AALDH1A1ADRB1LMNA
SCHEMBL7303819 0.78 PDE3B (0.46) PDE3BPDE3AABCB11MAOAADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5135932-A 2-HYDROXYPROPYLAMINO-ALKYL-BENZIMIDAZOLY-5-YL DERIVATIVES AND THEIR USE IN THE TREATMENT OF HEART DISEASE DR. KARL THOMAE GMBH (DE) 1992-08-04 US disclosed
EP-0400519-A1 2-Hydroxy-n-propylamines, medicaments containing these compounds and method for preparing them Dr. Karl Thomae GmbH (DE) 1990-12-05 EP disclosed