SCHEMBL7304744

SCHEMBL7304744

NC(=O)C(F)(F)C(O)C(CC1CCCCC1)NC(=O)OCc1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CTSB P07858 3/20 0.49
CTSL P07711 2/20 0.49
CTSS P25774 2/20 0.49
CTSK P43235 2/20 0.49
CASP1 P29466 1/20 0.46
REN P00797 3/20 0.44
ALDH1A1 P00352 1/20 0.43
TSHR P16473 1/20 0.42
EPHX1 P07099 1/20 0.42
HTRA1 Q92743 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7294910 0.92 CTSK (0.53) CTSBCTSLCTSSCTSKCASP1
SCHEMBL7427885 0.86 CTSB (0.49) CTSBCTSLCTSSCTSKCASP1
SCHEMBL7429221 0.86 CTSK (0.52) CTSBCTSLCTSSCTSKCASP1
SCHEMBL7434284 0.85 CTSK (0.51) CTSBCTSLCTSSCTSKCASP1
SCHEMBL7329100 0.85 CTSK (0.51) CTSBCTSLCTSSCTSKCASP1
SCHEMBL7427667 0.83 REN (0.49) CTSBCTSLCTSSCTSKREN
SCHEMBL9724730 0.82 TRPM8 (0.53) CTSBCTSLCTSSCTSKALDH1A1
SCHEMBL8759915 0.82 CTSB (0.55) CTSBCTSLCTSSCTSKCASP1
SCHEMBL7278761 0.81 REN (0.50) CTSBCTSLCTSSCTSKREN
SCHEMBL7293547 0.81 CTSB (0.54) CTSBCTSLCTSSCTSKCASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0368719-B1 Novel analogs of peptidase substrates MERRELL PHARMA INC (US) 1997-01-08 EP disclosed
US-5114927-A Hypotensive agents and inhibiting renin MERRELL DOW PHARMACEUTICALS INC. (US) 1992-05-19 US disclosed
EP-0371179-A1 Novel analogs of peptidase substrates MERRELL DOW PHARMACEUTICALS INC. (US) 1990-06-06 EP disclosed
EP-0356595-A1 Novel peptidase inhibitors MERRELL DOW PHARMACEUTICALS INC. (US) 1990-03-07 EP disclosed