SCHEMBL7310863

SCHEMBL7310863

CC(C)N1CCN(CCCN2CC(COS(C)(=O)=O)OC2=O)CC1

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
MAOB P27338 8/20 0.39
DAO P14920 1/20 0.34
HTR2B P41595 2/20 0.34
MAOA P21397 4/20 0.32
SLC6A4 P31645 1/20 0.31
HRH3 Q9Y5N1 1/20 0.31
DRD2 P14416 2/20 0.31
DRD3 P35462 2/20 0.31
KCNH2 Q12809 2/20 0.31
SLC2A1 P11166 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7316915 0.87 MAPK1 (0.45) MAPK1L3MBTL1
SCHEMBL7306386 0.85 MAPK1 (0.47) MAPK1L3MBTL1DRD2DRD3
SCHEMBL8858159 0.84 ITGB3 (0.34) MAPK1L3MBTL1HTR2B
SCHEMBL7306687 0.82 MAPK1 (0.35) MAPK1L3MBTL1HRH3
SCHEMBL7305151 0.81 MAPK1 (0.39) MAPK1L3MBTL1MAOAHRH3DRD2
SCHEMBL7308886 0.81 MAPK1 (0.49) MAPK1L3MBTL1DRD2DRD3
SCHEMBL8858107 0.81 KDM4E (0.33) MAPK1L3MBTL1HTR2B
SCHEMBL7314450 0.80 HTR7 (0.41) MAPK1L3MBTL1
SCHEMBL7227670 0.79 CHRM2 (0.41) MAPK1L3MBTL1
SCHEMBL7310668 0.79 MAPK1 (0.49) MAPK1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5776937-A Adhesion receptor antagonists MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1998-07-07 US disclosed
EP-0727425-A1 Adhesion receptor antagonists MERCK PATENT GmbH (DE) 1996-08-21 EP disclosed
EP-0711770-A1 Antagonists of adhesion receptors MERCK PATENT GmbH (DE) 1996-05-15 EP disclosed