SCHEMBL7305459

SCHEMBL7305459

CSCC[C@H](NCCC(c1ccccc1)c1ccccc1)C(N)=O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 1/20 0.48
MTNR1B P49286 1/20 0.48
CYP3A4 P08684 2/20 0.46
CYP1A2 P05177 2/20 0.46
CYP2D6 P10635 2/20 0.46
CYP2C19 P33261 2/20 0.46
CASR P41180 2/20 0.46
HTR1A P08908 2/20 0.46
ADORA3 P0DMS8 2/20 0.46
SLC6A2 P23975 2/20 0.46
SLC6A4 P31645 2/20 0.46
ADRA1A P35348 2/20 0.46
OPRM1 P35372 2/20 0.46
DRD3 P35462 2/20 0.46
SLC6A3 Q01959 2/20 0.46
KCNH2 Q12809 2/20 0.46
CHRM2 P08172 1/20 0.46
ADRA2A P08913 1/20 0.46
CHRM1 P11229 1/20 0.46
SMPD1 P17405 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7317844 0.90 GAA (0.43) MTNR1AMTNR1BLMNAMEN1ALDH1A1
SCHEMBL7313618 0.83 CA1 (0.47) FNTAFNTBGAAOPRK1ANPEP
SCHEMBL10764115 0.81 GGT1 (0.52) CYP2D6CYP2C19KMT2AFNTAFNTB
Hydrochloric Acid SCHEMBL11094927 0.80 GGT1 (0.51) CYP2D6CYP2C19MEN1KMT2AFNTA
SCHEMBL7303559 0.80 GAA (0.44) LMNAMEN1ALDH1A1KMT2ATSHR
SCHEMBL7319574 0.80 CASR (0.53) MTNR1AMTNR1BCYP3A4CYP1A2CYP2D6
SCHEMBL7265651 0.80 ANPEP (0.55) TSHRGAAANPEP
SCHEMBL7313416 0.79 MAPT (0.44) TSHRGAAANPEP
SCHEMBL7317918 0.78 CTSK (0.46) MTNR1AMTNR1BLMNAMEN1ALDH1A1
SCHEMBL9190837 0.77 TSHR (0.38) LMNAALDH1A1TSHRFNTAFNTB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1041064-A2 N-substituted alpha aminoacid amides as calcium channel modulators ELI LILLY AND COMPANY LIMITED (GB) 2000-10-04 EP disclosed
EP-0805147-A1 Novel N-substituted alpha aminoacid amides as calcium channel modulators LILLY INDUSTRIES LIMITED (GB) 1997-11-05 EP disclosed