SCHEMBL7306604

SCHEMBL7306604

CC(C)C[C@H](NC(c1ccccc1)c1ccccc1)C(=O)NC(=O)OC(C)(C)C

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.46
NPSR1 Q6W5P4 3/20 0.46
POLB P06746 2/20 0.46
RECQL P46063 2/20 0.46
ALDH1A1 P00352 1/20 0.46
CTSK P43235 7/20 0.46
CTSS P25774 3/20 0.46
CTSL P07711 2/20 0.46
CTSB P07858 1/20 0.44
REN P00797 2/20 0.44
MAPK1 P28482 2/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
AAK1 Q2M2I8 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7301520 0.84 CTSK (0.44) MAPTNPSR1POLBRECQLALDH1A1
SCHEMBL7304463 0.83 CYP1A2 (0.43) NPSR1ALDH1A1CTSKCTSSCTSL
SCHEMBL8083658 0.83 CTSK (0.46) MAPTNPSR1RECQLALDH1A1CTSK
SCHEMBL8083650 0.82 PPARG (0.45) MAPTALDH1A1CTSKCTSSCTSL
SCHEMBL7317017 0.82 CTSK (0.47) MAPTALDH1A1CTSKCTSSREN
SCHEMBL10630212 0.81 CTSK (0.57) MAPTNPSR1POLBRECQLALDH1A1
SCHEMBL7304711 0.81 CTSK (0.44) MAPTNPSR1RECQLALDH1A1CTSK
SCHEMBL7307182 0.81 CTSK (0.44) MAPTNPSR1RECQLALDH1A1CTSK
SCHEMBL7316620 0.79 CTSK (0.57) ALDH1A1CTSKCTSSCTSLCTSB
SCHEMBL8086793 0.79 KMT2A (0.52) NPSR1ALDH1A1CTSKCTSSCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1041064-A2 N-substituted alpha aminoacid amides as calcium channel modulators ELI LILLY AND COMPANY LIMITED (GB) 2000-10-04 EP disclosed
EP-0805147-A1 Novel N-substituted alpha aminoacid amides as calcium channel modulators LILLY INDUSTRIES LIMITED (GB) 1997-11-05 EP disclosed